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(2S)-2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
1-cyclopropyl-4-(4-phenyl-1,4-diazepane-1-carbonyl)pyrrolidin-2-one
1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-2-(propylsulfanyl)ethan-1-one
4-fluoro-2-hydroxy-N-[(1r,4r)-4-methoxycyclohexyl]benzamide
2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]acetamide
1-[(1S,5R)-6-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-(dimethylamino)-N-{2-[ethyl(methyl)amino]-2-methylpropyl}-2-(3-methylphenyl)acetamide
3-phenyl-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperazine
{1-[4-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
(2E)-N-{[3-methyl-7-(2-phenoxyacetyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
(1R,3S,5S)-8-(2,7-dimethylquinoline-4-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
(2R,6R)-1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]but-2-ynamide
N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylfuran-3-carboxamide
2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
N-[2-(3-methoxyphenyl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]ethyl]-N-methylpyridine-2-carboxamide
ethyl 5-(1H-indazole-3-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 3-(3-methylbutyl)-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]pyridine
9-[3-(2-fluorophenyl)propanoyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(4-fluorophenyl)methyl]-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decane
methyl 2-({5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}amino)benzoate
N-[(2,3-dimethoxyphenyl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-(4-chloro-1H-pyrazole-3-carbonyl)-3-[2-(2-methylphenyl)ethyl]piperidine
N-[(3R,4S)-4-cyclopropyl-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]pyrrolidin-3-yl]methanesulfonamide
methyl 3-({[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)propanoate
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[4-(morpholin-4-yl)butan-2-yl]acetamide
methyl 3-{[1-(cyclopropylmethyl)-5-(2,3-dimethylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-[(1H-1,2,3,4-tetrazol-5-ylmethyl)amino]pyridine-3-carboxamide
N-{2-[2-(pyridin-2-yl)ethyl]phenyl}thiomorpholine-4-carboxamide
2,3-dimethyl-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
3-[3-(1-methoxyethyl)phenyl]-5-(propan-2-yl)-1H-1,2,4-triazole
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[3-(thiomorpholin-4-ylmethyl)phenoxy]piperidin-1-yl}ethan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(6-ethyl-2-methylpyrimidin-4-yl)-N-methylpiperidin-4-amine
5-(propan-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,2-oxazole-3-carboxamide
(1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
dimethyl(3-{2-[1-(5,6,7,8-tetrahydroquinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-[3-(phenylamino)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[2-(benzenesulfonyl)ethyl]-1,4-oxazepan-5-one
2-(4-chloro-2-methylphenoxy)-1-{4-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propan-1-one
1,3-dimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
ethyl 5-(2,3-dimethylquinoxaline-6-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(3-methylbutyl)-8-(morpholine-4-sulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[(2,6-dimethoxyphenyl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1,2-oxazole-5-carboxamide
2-chloro-N-(2,3-dihydro-1H-inden-2-yl)-5-acetamido-N-methylbenzamide