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6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-[2-(3,4,5-trimethoxyphenyl)acetyl]-1,4-diazepan-2-one
1-benzyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(1R,2S)-2-phenylcyclohexyl]acetamide
2-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyridine-3-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
methyl 5-{[4-(methylsulfamoyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-3-(1H-imidazol-2-yl)piperidine
methyl 3-[(3S,4R)-4-(dimethylamino)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl]propanoate
4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-N,N-dimethylpiperazine-1-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
N-[2-(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
2-(2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)-1,2,3,4-tetrahydroisoquinoline
4-[(2-chloro-6-fluorophenyl)methyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
1-methyl-2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]azepane
(3R,4S)-4-[ethyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]oxolan-3-ol
1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
8-(6-methoxypyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-({4-[1-(furan-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-{1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
2-butyl-N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2,5-dihydro-1H-pyrrole-1-carboxamide
(3S,9aR)-3-(4-aminobutyl)-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-(cyclopropylmethyl)-1-methyl-4-(2-methylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2,4-difluorophenyl)-3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)benzamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}thiomorpholine
1-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}piperidin-4-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxane-2-carboxamide
N-benzyl-1-{2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-(pyrrolidin-3-yl)benzamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
5-{2-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
(3S,4S)-N-[3-(benzyloxy)phenyl]-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
2-[(2-cyclopropyl-1H-imidazol-1-yl)methyl]adamantan-2-ol
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,3-dimethylcyclohexan-1-amine
N-{[1-(2-cyclopentylacetyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
1,7-dimethyl-2-(4-methyl-2-phenylpiperazine-1-carbonyl)-1H-indole
N-(4-{4-[4-ethyl-1-(2-methylprop-2-en-1-yl)-2,5-dioxoimidazolidin-4-yl]piperidine-1-carbonyl}phenyl)acetamide
methyl 3-[2-(2,5-difluorophenyl)acetyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl 1-[(3S,5S)-1-(3-methylbut-2-en-1-yl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(thiophen-3-ylmethyl)amino]methyl}piperidin-2-one
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
2-{[2-(2,5-dimethylphenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-5-methyl-N-(2-phenylethyl)thieno[2,3-d]pyrimidin-4-amine
2-(4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
1-{3-[3-(3-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
2,4-dimethyl-N-[2-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
methyl 3-[(3-cyclohexylpropanamido)methyl]-5-[2-(1,3-thiazol-4-yl)acetamido]benzoate