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methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(4-methyl-1,3-oxazole-5-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(2-methoxy-5-methylphenyl)pyrimidine
5,5-dimethyl-3-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1,3-oxazolidine-2,4-dione
N-[(2R,3R)-2-hydroxy-1'-[(3-hydroxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
(4aR,8aS)-1-(3-ethoxypropyl)-6-[(3-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
(2R)-2-cyclohexyl-2-hydroxy-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2,6-dimethoxy-3-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}pyridine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
1-{9-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-3-azaspiro[5.5]undecan-3-yl}pentan-1-one
3-[(3-methoxyphenyl)methyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5S)-5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]pyrrolidin-3-ol
2-chloro-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]quinoxaline-5-carboxamide
5-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
6-(3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-9H-purine
2-{[2-(phenylamino)pyrimidin-5-yl]formamido}-N-(propan-2-yl)acetamide
methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})[3-(pyrrolidin-1-yl)propyl]amine
N1-ethyl-N2-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1,2-dicarboxamide
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-ethyl-N-(2-hydroxyethyl)acetamide
1-acetyl-N-[3-(3-chlorophenyl)phenyl]piperidine-4-carboxamide
(3S,9aR)-3-ethyl-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,7aR)-1-[(2-fluorophenyl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-[(3-methoxyphenyl)methyl]-1,2-oxazole-5-carbonyl}-4-phenylazepane
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
2,5-dimethoxy-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
3-(2-fluoro-5-methoxyphenyl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
2-methoxy-4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
4-{1-[1-(furan-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-(4-ethylpiperazin-1-yl)-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
3,5-dimethyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2-oxazole-4-sulfonamide
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-(thiophen-3-yl)propan-1-one
6-{7-methyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}-1,2-dihydropyridin-2-one
N-[2-({3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)quinolin-5-yl]acetamide
8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
N-[(8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]oxane-4-carboxamide
5,7-dimethyl-N-[2-(4-methylpiperazin-1-yl)butyl]pyrido[2,3-d]pyrimidin-4-amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethyl-4-phenylpyrimidine-5-carboxamide
4-(cyclopropylmethyl)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
4,6-dimethyl-2-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-3-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
3-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-methylpropanamide
4-(2,3-dihydro-1H-inden-2-yl)-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
2-(dimethylamino)-8-(isoquinolin-5-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(oxolan-2-ylmethyl)cyclopropane-1-carboxamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-butylpropanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
2-[(isoquinolin-5-yloxy)methyl]-N-[1-(5-methylpyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide