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4-{3-methyl-5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
3-hydroxy-5-(2-methoxyquinolin-3-yl)benzoic acid
1-{[5-(3,6-dimethylpyrazin-2-yl)-2-hydroxyphenyl]methyl}piperidin-3-ol
1-(4-{[2-(2-methoxynaphthalen-1-yl)ethyl]amino}piperidin-1-yl)-2-methylpropan-1-one
N-{2-[4-({[(3,4-dimethylphenyl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}methanesulfonamide
methyl 3-[(2-methoxyphenyl)methyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-methyl-2-({[2-methyl-1-(pyridin-2-yl)propyl]amino}methyl)quinolin-4-ol
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-3-yl)acetamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(thiophene-3-carbonyl)pyrrolidin-3-yl]acetamide
1-[1-(propan-2-yl)piperidine-4-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-2-[4-(pyrrolidine-1-carbonyl)morpholin-3-yl]acetamide
(2E)-1-[(4aR,8aS)-6-acetyl-decahydro-1,6-naphthyridin-1-yl]-3-(3,4-difluorophenyl)prop-2-en-1-one
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)butan-1-one
N-[(2,3-dimethoxyphenyl)methyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyridin-3-yl)acetamide
N-(2,3-dihydro-1H-inden-2-yl)-1-{4-[(dimethylsulfamoyl)amino]phenyl}piperidin-4-amine
2-[cyclohexyl(methyl)amino]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-3-carboxamide
1-[(3S)-3-(dimethylamino)azepan-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-ethyl-2-[(3S)-3-hydroxypyrrolidin-1-yl]-N-(2-methoxyethyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
ethyl 1-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidine-4-carboxylate
2-(aminomethyl)-N-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)piperidine-1-carboxamide
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
1-{1-[1-(2-ethylpyridine-4-carbonyl)piperidin-4-yl]ethyl}-4-methylpiperazine
3-cyclopropyl-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[3-(1H-imidazol-1-yl)propyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidine-2-carboxamide
(2E)-N-({7-[4-(4-fluorophenyl)-4-oxobutanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-benzyl-5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]phenoxy}-N-methylacetamide
4-{4-[(1,3-dihydroxypropan-2-yl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-methyl-1,3-benzothiazole-6-sulfonamide
1-[6-(2-methylpyrrolidin-1-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyridine-3-carboxamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-N-[(4-fluorophenyl)methyl]propanamide
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
N-ethyl-5-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]pyrimidin-2-amine
N,1-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]pyrimidin-4-amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}benzamide
2-[1-cyclopentyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(naphthalen-1-ylmethyl)acetamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(morpholin-4-yl)cyclohexane-1-carboxamide
3-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-6-phenylpyridazine
1-(1-benzylpyrrolidin-3-yl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
5-methoxy-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-4-oxo-1,4-dihydropyridine-2-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid