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2-butyl-4-methyl-3-oxo-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-(1-hydroxybutan-2-yl)-N-(pyridin-4-ylmethyl)acetamide
9-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-[(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]piperazine
6-(4-ethylphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-[3-(pyridin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
(2S,4S)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-(5-methylthiophene-2-amido)pyrrolidine-2-carboxamide
3-[(4-methoxyphenyl)methyl]-8-[3-(5-methylfuran-2-yl)butyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(2,5-dimethylphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(5-chloro-1H-indol-2-yl)methyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
6-{4-[(2-methoxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}pyridine-2-carbonitrile
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-methoxypiperidine
6-(1-methyl-1H-imidazol-2-yl)-N-[2-(morpholin-4-yl)ethyl]pyridazin-3-amine
N-[(8-{[2-(furan-2-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]-1-methyl-1H-pyrazole-5-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2,3-dihydro-1,4-benzodioxine-5-carboxamide
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-(pyridin-2-yl)pyrimidine
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
3-(3,4-dimethoxybenzoyl)-1-[(5-ethylfuran-2-yl)methyl]piperidine
(3S,4R)-1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-2-amine
2-amino-4-(4-methyl-1,3-thiazol-2-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
4-chloro-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}aniline
5-methanesulfonyl-1'-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-6-methylpyridine
4-cyclopropyl-6-{3-[(methylsulfanyl)methyl]piperidin-1-yl}pyrimidine
5-(3-methoxyphenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(benzyloxy)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
4-(2,5-dimethoxyphenyl)-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[3-(cyclopentyloxy)phenyl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
5-[({1-[3-(3-methylphenyl)phenyl]piperidin-4-yl}amino)methyl]pyrrolidin-2-one
ethyl 4-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
N-[2-(dimethylsulfamoyl)ethyl]-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
6-(4-methylpiperazin-1-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-2,1,3-benzoxadiazole
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-(pyrazin-2-yl)-2-({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)acetamide
N-ethyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(pyridin-4-ylmethyl)acetamide
2-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
1-[(2-fluorophenyl)methyl]-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-2-amine
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]propanamide
5-acetyl-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-3-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidin-3-amine
[(3-{[1-(5-chloro-3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
2-(5-cyclopropyl-1H-pyrazol-3-yl)-7-(4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(4-hydroxypiperidin-1-yl)-2-[4-(4-{[2-(naphthalen-1-yl)ethyl]amino}piperidin-1-yl)phenyl]ethan-1-one