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3-{[2-(1H-indol-3-yl)ethyl]carbamoyl}pyrazine-2-carboxylic acid
3-[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-3,4-dihydroquinazolin-4-one
6,7-dimethoxy-2-[3-(1H-pyrrol-1-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{6-methoxy-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrrolidine-2,5-dione
4-{6,7-dimethoxy-1-methyl-1H,4H-indeno[1,2-c]pyrazole-3-amido}benzoic acid
N-(2,3-dihydro-1H-inden-2-yl)-2-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]acetamide
(2S)-N-cyclopentyl-2-[2-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)acetamido]-4-(methylsulfanyl)butanamide
N-[2-(1H-indol-3-yl)ethyl]-N'-(1H-indol-6-yl)ethanediamide
N-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyethyl)-4-oxo-3,4-dihydroquinazoline-2-carboxamide
(1S,9R)-6-oxo-N-(4-oxo-3,4,5,6,7,8-hexahydroquinazolin-2-yl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carboximidamide
N-{2-[(1-methyl-1H-indol-2-yl)formamido]ethyl}pyridine-3-carboxamide
2-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-(3,4,5-trimethoxyphenyl)acetamide
methyl 3-{[4-(2,3-dimethoxyphenyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]amino}propanoate
9-oxo-N-(pyridin-2-ylmethyl)-1H,2H,3H,9H-pyrrolo[2,1-b]quinazoline-6-carboxamide
2-N-(3,4-dimethoxyphenyl)-6-N-(2-methoxyethyl)-9H-purine-2,6-diamine
1-benzyl-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrrolidine-2,5-dione
3-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)-N-(6-methylheptan-2-yl)propanamide
1-(2,3-dimethoxybenzoyl)-1H,2H,3H,5H-imidazolidino[1,2-b]isoquinolin-5-one
methyl 2-{11,13-dimethyl-6-oxo-8-oxa-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-5-yl}acetate
(2S)-2-[2-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)acetamido]-N-(2-hydroxyethyl)-4-(methylsulfanyl)butanamide
3-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)-N-(3,4,5-trimethoxyphenyl)propanamide
2-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-(3-acetamidophenyl)acetamide
N-(3-methylbutyl)-2-(pyridin-2-yl)quinoline-4-carboxamide
(5s,7s)-2-(7-methoxy-1H-indol-3-yl)-5,7-dimethyl-1,3-diazatricyclo[3.3.1.13,7]decan-6-one
5-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-{4-methoxy-6-methyl-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]isoquinolin-9-yl}furan-2-carboxamide
(2E)-3-(2H-1,3-benzodioxol-5-yl)-N-cyclopropyl-N-(1H-indol-4-ylmethyl)prop-2-enamide
6-N-(2H-1,3-benzodioxol-5-ylmethyl)-9H-purine-2,6-diamine
(5s,7s)-2,2,5-trimethyl-7-phenyl-1,3-diazatricyclo[3.3.1.13,7]decan-6-ol
(2S)-2-[2-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)acetamido]-3-methyl-N-(1,3-thiazol-2-yl)pentanamide
2-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-phenylacetamide
N-(2,4-dimethoxyphenyl)-12-oxo-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide
1-(4-fluorophenyl)-N-{4-methoxy-6-methyl-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]isoquinolin-9-yl}-4-oxo-1,4-dihydropyridazine-3-carboxamide
12-oxo-N-phenyl-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide
(2S)-2-[2-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)acetamido]-N-(4-methyl-1,3-thiazol-2-yl)-4-(methylsulfanyl)butanamide
methyl 4-{[4-(3-methoxyphenyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]amino}butanoate
N-(3-methoxypropyl)-12-oxo-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide
(5r,7r)-2-(1H-indol-4-yl)-5,7-dimethyl-1,3-diazatricyclo[3.3.1.13,7]decane
methyl (2S)-2-{[4-(3,5-dimethoxyphenyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]amino}-3-phenylpropanoate
N-(2H-1,3-benzodioxol-5-ylmethyl)-6,7-dimethoxy-1-methyl-1H,4H-indeno[1,2-c]pyrazole-3-carboxamide
(1s,5s)-3,7-bis(1H-indole-3-carbonyl)-1,5-dimethyl-3,7-diazabicyclo[3.3.1]nonan-9-ol
4-[6-(4-oxo-3,4-dihydroquinazolin-3-yl)hexanamido]benzamide
2-[(5-hydroxy-2,2-dimethyl-4-oxo-3,4-dihydro-2H-1-benzopyran-7-yl)oxy]-N-(1H-indol-6-yl)acetamide
N-(3-methylbutyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}-2-(5-bromofuran-2-yl)-1,3-oxazole-4-carbonitrile
2-[(4,6-dimethylpyrimidin-2-yl)amino]-3-(1H-indol-3-yl)propanoic acid
(2E)-3-(4-methoxyphenyl)-N-(quinolin-5-yl)prop-2-enamide
4-[(4,5-dimethoxy-3-oxo-1,3-dihydro-2-benzofuran-1-yl)amino]benzamide
4-(1H-indol-3-yl)-N-{2-[(1-methyl-1H-indol-2-yl)formamido]ethyl}butanamide
methyl (2S)-2-{[4-(2,3-dimethoxyphenyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]amino}propanoate
N-(6-methylheptan-2-yl)-9-oxo-1H,2H,3H,9H-pyrrolo[2,1-b]quinazoline-6-carboxamide