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N-(3-acetylphenyl)-2-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]acetamide
N-cyclopropyl-3-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]propanamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]propanamide
2-(5,7-dimethoxy-4-methyl-2-oxo-2H-chromen-3-yl)-N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]acetamide
(5s,7s)-2-(6-chloro-1H-indol-3-yl)-5,7-dimethyl-1,3-diazatricyclo[3.3.1.13,7]decan-6-one
2-(7-methoxy-1H-indol-1-yl)-N-(propan-2-yl)acetamide
N-{4-methoxy-6-methyl-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]isoquinolin-9-yl}-4-(3-methyl-4-oxo-3,4-dihydrophthalazin-1-yl)benzamide
methyl 4-{2-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]acetamido}butanoate
4-[6-(2,4-dioxo-1,2,3,4-tetrahydroquinazolin-3-yl)hexanamido]benzamide
1,4-dimethyl (2S)-2-{[4-(2-methoxyphenyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]amino}butanedioate
methyl (2S)-2-[2-(7-methoxy-1H-indol-1-yl)acetamido]-4-(methylsulfanyl)butanoate
N-{2-[(1-methyl-1H-indol-2-yl)formamido]ethyl}-1H-indole-4-carboxamide
4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-(pyridin-3-yl)quinoline
4-[2-(7,8-dimethoxy-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]benzamide
2-[4-(benzyloxy)phenyl]-5-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-1,3-oxazole-4-carbonitrile
(3S)-3-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-(furan-2-ylmethyl)-N-{4-methoxy-6-methyl-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]isoquinolin-9-yl}-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
N-cyclopropyl-N-(1H-indol-6-ylmethyl)-2-methoxyacetamide
N-{4-methoxy-6-methyl-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]isoquinolin-9-yl}quinoline-2-carboxamide
N-{4-methoxy-6-methyl-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]isoquinolin-9-yl}-3-phenylpropanamide
(5s,7s)-2-(1H-indol-6-yl)-5,7-dimethyl-1,3-diazatricyclo[3.3.1.13,7]decan-6-ol
N-[2-(1H-indol-3-yl)ethyl]-2-(7-methoxy-1H-indol-1-yl)acetamide
3-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-(3-phenylpropyl)propanamide
3-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)-N-(1H-indol-5-yl)propanamide
3-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)-N-[2-(4-methoxyphenyl)ethyl]propanamide
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-[(phenylcarbamoyl)methyl]-1,2,4-oxadiazole-5-carboxamide
3-[(4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxoimidazolidin-4-yl]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]propanamide
N-(2-methoxyphenyl)-12-oxo-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide
3-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)-N-[3-(dimethylamino)propyl]propanamide
ethyl 4-{6,7-dimethoxy-1-methyl-1H,4H-indeno[1,2-c]pyrazole-3-amido}benzoate
2-(4-chlorophenyl)-5-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-1,3-oxazole-4-carbonitrile
3-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-(2-methylpropyl)propanamide
N-benzyl-3-[(3S)-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-3-yl]-N-methylpropanamide
methyl (2S)-4-(methylsulfanyl)-2-{[2-(pyridin-2-yl)quinolin-4-yl]formamido}butanoate
3-(2-methoxyethyl)-N-methyl-4-oxo-3,4-dihydroquinazoline-2-carboxamide
1-benzyl-3-{6-methoxy-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrrolidine-2,5-dione
(2E)-3-(2-methoxyphenyl)-N-(quinolin-5-yl)prop-2-enamide
(1s,5s)-1,5-dimethyl-9-oxo-3,7-diazabicyclo[3.3.1]nonane-3,7-dicarbaldehyde
(furan-2-ylmethyl)({2-[4-(4-methoxyphenyl)-2,2-dimethyloxan-4-yl]ethyl})amine
(2S)-2-[2-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)acetamido]-3-methyl-N-(pyridin-4-ylmethyl)pentanamide
(2R)-1-(3-{4-methyl-7-[(2-methylprop-2-en-1-yl)oxy]-2-oxo-2H-chromen-3-yl}propanoyl)pyrrolidine-2-carboxamide
1-{9-oxo-1H,2H,3H,9H-pyrrolo[2,1-b]quinazoline-6-carbonyl}piperidine-4-carboxamide
3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-1-(3,4,5-trimethoxyphenyl)pyrrolidine-2,5-dione
(2S)-2-[2-(5-methoxy-1H-indol-1-yl)acetamido]-3-methylbutanoic acid
methyl 6,7-dimethoxy-1-methyl-1H,4H-indeno[1,2-c]pyrazole-3-carboxylate
2-(5-benzamido-1H-indol-3-yl)-2-[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]acetic acid
(2S)-2-[2-(6,7-dimethoxy-4-oxo-3,4-dihydroquinazolin-3-yl)acetamido]-N-(2-hydroxyphenyl)-4-(methylsulfanyl)butanamide
(3S)-3-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
5-(4-chlorophenyl)-N-{4-methoxy-6-methyl-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]isoquinolin-9-yl}furan-2-carboxamide
2-(3-methoxyphenyl)-5-[(1S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]-1,3-oxazole-4-carbonitrile