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3-{[(1S)-1-{[(2S)-4-methyl-1-[(2S)-2-{[(1S)-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]-2-phenylethyl]carbamoyl}pyrrolidin-1-yl]-1-oxopentan-2-yl]carbamoyl}ethyl]carbamoyl}propanoic acid
tert-butyl N-[(1S)-5-acetamido-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]pentyl]carbamate
(4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-5-amino-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]pentyl]carbamoyl}-2-methylpropyl]carbamoyl}-2-methylpropyl]carbamoyl}-3-carboxypropyl]carbamoyl}-4-acetamidobutanoic acid
(4S)-4-{[(1S,2R)-1-{[(1S)-2-carboxy-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]ethyl]carbamoyl}-2-hydroxypropyl]carbamoyl}-4-[(2S)-2-acetamido-3-methylbutanamido]butanoic acid
(4S)-4-[(2S)-2-[(2S)-2-{[(benzyloxy)carbonyl]amino}-4-methylpentanamido]-4-methylpentanamido]-4-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]butanoic acid
(2S)-N-[(1S)-5-amino-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]butyl]carbamoyl}-3-methylbutyl]carbamoyl}pentyl]-2-[(2S)-6-amino-2-acetamidohexanamido]pentanediamide
benzyl N-[(1S)-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]butyl]carbamoyl}-2-methylpropyl]carbamoyl}-2-methylpropyl]carbamate
benzyl N-[(1S)-1-{[(1S)-5-amino-1-{[(1S)-4-carbamimidamido-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]butyl]carbamoyl}pentyl]carbamoyl}ethyl]carbamate
tert-butyl N-[(1S)-2-hydroxy-1-{[(1S)-1-{[(1S)-3-methyl-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]butyl]carbamoyl}-2-phenylethyl]carbamoyl}ethyl]carbamate
(4S)-4-{[(1S)-5-amino-1-[(4-methyl-2-oxo-2H-chromen-7-yl)carbamoyl]pentyl]carbamoyl}-4-[(2S)-2-{[(benzyloxy)carbonyl]amino}-3-(1H-imidazol-4-yl)propanamido]butanoic acid
(4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-4-carbamimidamido-1-carbamoylbutyl]carbamoyl}butyl]carbamoyl}-5-[(2,4-dinitrophenyl)amino]pentyl]carbamoyl}butyl]carbamoyl}-2-phenylethyl]carbamoyl}-3-carboxypropyl]carbamoyl}ethyl]carbamoyl}-2-carboxyethyl]carbamoyl}-3-methylbutyl]carbamoyl}-2-carbamoylethyl]carbamoyl}-2-methylpropyl]carbamoyl}-4-[(2S)-3-hydroxy-2-[2-(4-methoxy-2-oxo-2H-chromen-8-yl)acetamido]propanamido]butanoic acid
(2S)-2-[(2S)-2-[(2S)-2-amino-5-carbamimidamidopentanamido]-5-carbamimidamidopentanamido]-N-({[(1S)-1-{[(1S)-1-{[(1S,2S)-1-{[(1S)-1-{[(1S,2S)-1-{[(1S)-1-{[(1S,2R)-1-{[(1S,2R)-1-{[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(1S)-4-carbamimidamido-1-carbamoylbutyl]carbamoyl}butyl]carbamoyl}-5-[(2,4-dinitrophenyl)amino]pentyl]carbamoyl}-2-methylbutyl]carbamoyl}-2-methylbutyl]carbamoyl}-2-methylpropyl]carbamoyl}-2-hydroxypropyl]carbamoyl}ethyl]carbamoyl}-2-methylbutyl]carbamoyl}-2-methylpropyl]carbamoyl}-2-methylpropyl]carbamoyl}methyl)-6-[2-(4-methoxy-2-oxo-2H-chromen-8-yl)acetamido]hexanamide
(4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-5-amino-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-carbamoyl-5-[(2,4-dinitrophenyl)amino]pentyl]carbamoyl}-2-phenylethyl]carbamoyl}-2-methylpropyl]carbamoyl}-3-methylbutyl]carbamoyl}pentyl]carbamoyl}-3-carboxypropyl]carbamoyl}-2-(1H-imidazol-4-yl)ethyl]carbamoyl}-2-(1H-imidazol-4-yl)ethyl]carbamoyl}-2-methylpropyl]carbamoyl}-4-[(2S)-3-(4-hydroxyphenyl)-2-[2-(7-methoxy-2-oxo-2H-chromen-4-yl)acetamido]propanamido]butanoic acid
(3S)-3-amino-1-chloro-5-methylhexan-2-one
benzyl N-({[(1S)-1-{[(2S)-4-chloro-3-oxo-1-phenylbutan-2-yl]carbamoyl}-3-methylbutyl]carbamoyl}methyl)carbamate
benzyl N-[(1S)-1-{[(2S)-4-chloro-3-oxobutan-2-yl]carbamoyl}-2-phenylethyl]carbamate
benzyl N-[(1S)-1-{[(2S)-4-chloro-3-oxo-1-phenylbutan-2-yl]carbamoyl}-2-phenylethyl]carbamate
(2S)-N-{[(3-chloro-2-oxopropyl)carbamoyl]methyl}-2-acetamido-3-(4-hydroxyphenyl)propanamide
methyl 3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(2S)-4-chloro-3-oxobutan-2-yl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}ethyl]carbamoyl}propanoate
benzyl (2S)-2-{[(1S)-1-{[(1S)-1-{[(2S)-4-chloro-3-oxobutan-2-yl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]carbamoyl}pyrrolidine-1-carboxylate
5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d]imidazolidin-4-yl]-N-{6-[(2S)-2-{[(1S)-1-{[(1S)-1-{[(2S)-4-chloro-3-oxobutan-2-yl]carbamoyl}-2-phenylethyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]carbamoyl}pyrrolidin-1-yl]-6-oxohexyl}pentanamide
methyl 3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(3S)-1-chloro-4-methyl-2-oxopentan-3-yl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}ethyl]carbamoyl}propanoate
(2S)-1-[(2S)-2-[(2S)-2-aminopropanamido]propanoyl]-N-[(3S)-1-chloro-4-methyl-2-oxopentan-3-yl]pyrrolidine-2-carboxamide
(2S)-2-[(2S)-2-aminopropanamido]-N-[(2S)-4-chloro-3-oxo-1-phenylbutan-2-yl]propanamide
5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d]imidazolidin-4-yl]-N-[(1S)-1-{[(1S)-1-{[(2S)-4-chloro-3-oxo-1-phenylbutan-2-yl]carbamoyl}ethyl]carbamoyl}ethyl]pentanamide
3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(2S)-4-chloro-3-oxo-1-phenylbutan-2-yl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}ethyl]carbamoyl}propanoic acid
(2S)-N-[(3S)-7-amino-1-chloro-2-oxoheptan-3-yl]-2-[(2R)-2-amino-3-methylbutanamido]-4-methylpentanamide
methyl (3S)-3-[(2S)-2-[(2S)-2-{[(benzyloxy)carbonyl]amino}propanamido]propanamido]-5-chloro-4-oxopentanoate
methyl (3S)-3-[(2S)-2-[(2S)-2-(6-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d]imidazolidin-4-yl]pentanamido}hexanamido)propanamido]propanamido]-5-chloro-4-oxopentanoate
methyl 3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(2S)-4-chloro-3-oxo-1-phenylbutan-2-yl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}-3-methylbutyl]carbamoyl}propanoate
tert-butyl N-[(1S)-1-{[(1S)-4-carbamimidamido-1-{[(3S)-6-carbamimidamido-1-chloro-2-oxohexan-3-yl]carbamoyl}butyl]carbamoyl}-3-methylbutyl]carbamate
methyl 3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(3S)-1-chloro-5-methyl-2-oxohexan-3-yl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}-2-(1H-indol-3-yl)ethyl]carbamoyl}propanoate
methyl 3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(2S)-4-chloro-1-(1H-indol-3-yl)-3-oxobutan-2-yl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}ethyl]carbamoyl}propanoate
(2S)-2-amino-4-(2-hydroxycarbamimidamido)butanoic acid
tert-butyl N-[(2R)-1-[(2S)-2-{[(R)-(4-carbamimidoylphenyl)(diphenoxyphosphoryl)methyl]carbamoyl}pyrrolidin-1-yl]-1-oxo-3-phenylpropan-2-yl]carbamate
methyl 3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(1R)-1-(diphenoxyphosphoryl)-2-methylpropyl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}ethyl]carbamoyl}propanoate
methyl 3-{[(1S)-1-{[(1S)-1-{[(1R)-1-(diphenoxyphosphoryl)-2-phenylethyl]carbamoyl}ethyl]carbamoyl}ethyl]carbamoyl}propanoate
diphenyl [(1R)-1-[(2S)-2-[(2S)-2-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d]imidazolidin-4-yl]pentanamido}propanamido]propanamido]-2-phenylethyl]phosphonate
methyl 3-{[(1S)-1-{[(2S)-1-[(2S)-2-{[(1R)-1-(diphenoxyphosphoryl)-2-phenylethyl]carbamoyl}pyrrolidin-1-yl]-1-oxopropan-2-yl]carbamoyl}ethyl]carbamoyl}propanoate
(3S)-3-{[(1S)-1-{[(R)-(4-carbamimidoylphenyl)(diphenoxyphosphoryl)methyl]carbamoyl}-2-phenylethyl]carbamoyl}-3-[(2S)-2-acetamido-3-(1H-imidazol-4-yl)propanamido]propanoic acid
(3S)-3-{[(1S)-1-{[(R)-(4-carbamimidoylphenyl)(diphenoxyphosphoryl)methyl]carbamoyl}-2-phenylethyl]carbamoyl}-3-[(2S)-2-acetamidohexanamido]propanoic acid
diphenyl [(2R)-1-[(2S)-2-aminopropanoyl]piperidin-2-yl]phosphonate
methyl (2S,3S)-2-[(2S)-2-[(4S)-4-[(2S,3S)-2-[(2S)-2-{[(tert-butoxy)carbonyl]amino}-3-methylbutanamido]-3-methylpentanamido]-2,2-difluoro-3-oxopentanamido]-3-methylbutanamido]-3-methylpentanoate
(3S)-3-amino-1-diazo-5-methylhexan-2-one
benzyl N-[(1S)-1-{[(2S)-4-($l^{5},-diazynylidene)-3-oxo-1-phenylbutan-2-yl]carbamoyl}-2-phenylethyl]carbamate
benzyl N-[(1S)-1-{[(2S)-4-($l^{5},-diazynylidene)-3-oxobutan-2-yl]carbamoyl}-2-phenylethyl]carbamate
2-amino-N-[(2S)-4-($l^{5},-diazynylidene)-3-oxo-1-phenylbutan-2-yl]acetamide
benzyl N-[(1S)-1-{[(1S)-1-{[(2S)-1-(4-hydroxyphenyl)-4-($l^{5},-diazynylidene)-3-oxobutan-2-yl]carbamoyl}-3-methylbutyl]carbamoyl}-3-methylbutyl]carbamate
benzyl N-[(1S)-2-(4-hydroxyphenyl)-1-{[(2S)-4-($l^{5},-diazynylidene)-3-oxobutan-2-yl]carbamoyl}ethyl]carbamate