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N-(5-carbamimidamido-1-{2-[(carbamoylmethyl)carbamoyl]pyrrolidin-1-yl}-1-oxopentan-2-yl)-2-{2-[2-(3-hydroxy-2-{2-[3-(1H-imidazol-4-yl)-2-[(5-oxopyrrolidin-2-yl)formamido]propanamido]-3-(1H-indol-3-yl)propanamido}propanamido)-3-(4-hydroxyphenyl)propanamido]acetamido}-4-methylpentanamide
N-(5-carbamimidamido-1-{2-[(carbamoylmethyl)carbamoyl]pyrrolidin-1-yl}-1-oxopentan-2-yl)-2-{2-[2-(3-hydroxy-2-{2-[3-(1H-imidazol-5-yl)-2-[(5-oxopyrrolidin-2-yl)formamido]propanamido]-3-(1H-indol-3-yl)propanamido}propanamido)-3-(4-hydroxyphenyl)propanamido]propanamido}-4-methylpentanamide
N-(5-carbamimidamido-1-{2-[(carbamoylmethyl)carbamoyl]pyrrolidin-1-yl}-1-oxopentan-2-yl)-2-[2-(2-{3-hydroxy-2-[3-(1H-indol-3-yl)-2-{2-[(5-oxopyrrolidin-2-yl)formamido]-3-phenylpropanamido}propanamido]propanamido}-3-(4-hydroxyphenyl)propanamido)-3-(1H-indol-3-yl)propanamido]-4-methylpentanamide
1-[5-carbamimidamido-2-(2-{2-[2-(3-hydroxy-2-{2-[3-(1H-imidazol-5-yl)-2-[(5-oxopyrrolidin-2-yl)formamido]propanamido]-3-(1H-indol-3-yl)propanamido}propanamido)-3-(4-hydroxyphenyl)propanamido]acetamido}-4-methylpentanamido)pentanoyl]-N-ethylpyrrolidine-2-carboxamide
1-[5-carbamimidamido-2-(2-{2-[2-(3-hydroxy-2-{2-[3-(1H-imidazol-5-yl)-2-[(5-oxopyrrolidin-2-yl)formamido]propanamido]-3-(1H-indol-3-yl)propanamido}propanamido)-3-(4-hydroxyphenyl)propanamido]propanamido}-4-methylpentanamido)pentanoyl]-N-ethylpyrrolidine-2-carboxamide
1-[5-carbamimidamido-2-(2-{2-[2-(3-hydroxy-2-{2-[3-(1H-imidazol-4-yl)-2-[(5-oxopyrrolidin-2-yl)formamido]propanamido]-3-(1H-indol-3-yl)propanamido}propanamido)-3-(4-hydroxyphenyl)propanamido]-3-(1H-indol-3-yl)propanamido}-4-methylpentanamido)pentanoyl]-N-ethylpyrrolidine-2-carboxamide
4-[2-(2-{2-[3-(acetyloxy)-2-acetamidopropanamido]-3-(4-hydroxyphenyl)propanamido}-3-hydroxypropanamido)-4-(methylsulfanyl)butanamido]-4-{[1-({1-[(1-{[1-({[(6-amino-1-{2-[(1-carbamoyl-2-methylpropyl)carbamoyl]pyrrolidin-1-yl}-1-oxohexan-2-yl)carbamoyl]methyl}carbamoyl)-2-(1H-indol-3-yl)ethyl]carbamoyl}-4-carbamimidamidobutyl)carbamoyl]-2-phenylethyl}carbamoyl)-2-(1H-imidazol-5-yl)ethyl]carbamoyl}butanoic acid
3-{2-[2-(2-{2-[2-(2-{2-[2-amino-3-(4-hydroxyphenyl)propanamido]-3-methylbutanamido}-4-(methylsulfanyl)butanamido)acetamido]-3-(1H-imidazol-4-yl)propanamido}-3-phenylpropanamido)-5-carbamimidamidopentanamido]-3-(1H-indol-3-yl)propanamido}-3-{[4-carbamimidamido-1-({1-[(carboxymethyl)carbamoyl]-2-phenylethyl}carbamoyl)butyl]carbamoyl}propanoic acid
4-[2-(2-amino-3-hydroxypropanamido)-4-(methylsulfanyl)butanamido]-4-{[1-({4-carbamimidamido-1-[({[1-carboxy-2-(1H-indol-3-yl)ethyl]carbamoyl}methyl)carbamoyl]butyl}carbamoyl)-2-methylpropyl]carbamoyl}butanoic acid
2-(2-{2-[(1-{2-[2-({1-[6-amino-2-(3-carbamoyl-2-{4-carbamoyl-2-[3-(4-hydroxyphenyl)-2-{4-methyl-2-[(5-oxopyrrolidin-2-yl)formamido]pentanamido}propanamido]butanamido}propanamido)hexanoyl]pyrrolidin-2-yl}formamido)-5-carbamimidamidopentanamido]-5-carbamimidamidopentanoyl}pyrrolidin-2-yl)formamido]-3-(4-hydroxyphenyl)propanamido}-3-methylpentanamido)-4-methylpentanoic acid
4-({1-[(6-amino-1-{2-[(4-carbamimidamido-1-{[5-carbamimidamido-1-(2-{[1-({1-[(1-carboxy-2-methylbutyl)carbamoyl]-2-methylbutyl}carbamoyl)-2-(1H-indol-3-yl)ethyl]carbamoyl}pyrrolidin-1-yl)-1-oxopentan-2-yl]carbamoyl}butyl)carbamoyl]pyrrolidin-1-yl}-1-oxohexan-2-yl)carbamoyl]-2-carbamoylethyl}carbamoyl)-4-[3-(4-hydroxyphenyl)-2-{4-methyl-2-[(5-oxopyrrolidin-2-yl)formamido]pentanamido}propanamido]butanoic acid
6-amino-2-(3-carbamoyl-2-{4-carboxy-2-[3-(4-hydroxyphenyl)-2-{4-methyl-2-[(5-oxopyrrolidin-2-yl)formamido]pentanamido}propanamido]butanamido}propanamido)hexanoic acid
2-{2-[2-({1-[2-(2-amino-5-carbamimidamidopentanamido)-5-carbamimidamidopentanoyl]pyrrolidin-2-yl}formamido)-3-(4-hydroxyphenyl)propanamido]-3-methylpentanamido}-4-methylpentanoic acid
2-[2-(2-{2-[2-(2-amino-5-carbamimidamidopentanamido)-3-(4-hydroxyphenyl)propanamido]-4-methylpentanamido}acetamido)-3-(4-hydroxyphenyl)propanamido]-4-methylpentanoic acid
2-{2-[2-(2-{2-[2-(2-amino-5-carbamimidamidopentanamido)-3-(4-hydroxyphenyl)propanamido]-4-methylpentanamido}acetamido)-3-(4-hydroxyphenyl)propanamido]-4-methylpentanamido}pentanedioic acid
2-[2-(2-{2-[2-amino-2-(methanethioyl)acetamido]-3-(4-hydroxyphenyl)propanamido}-3-methylpentanamido)-3-hydroxybutanamido]-N-(1-{[({1-[(carbamoylmethyl)carbamoyl]-3-methylbutyl}carbamoyl)methyl]carbamoyl}-2-sulfanylethyl)butanediamide
2-({1-[19-amino-13-benzyl-10-(2-carbamoylethyl)-7-(carbamoylmethyl)-16-[(4-hydroxyphenyl)methyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carbonyl]pyrrolidin-2-yl}formamido)-5-carbamimidamido-N-(carbamoylmethyl)pentanamide
6-amino-2-({1-[19-amino-13-benzyl-10-(2-carbamoylethyl)-7-(carbamoylmethyl)-16-[(4-hydroxyphenyl)methyl]-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carbonyl]pyrrolidin-2-yl}formamido)-N-(carbamoylmethyl)hexanamide
2-({1-[5-benzyl-8-(2-carbamoylethyl)-11-(carbamoylmethyl)-2-[(4-hydroxyphenyl)methyl]-3,6,9,12,20-pentaoxo-1,4,7,10,13-pentaazacycloicosane-14-carbonyl]pyrrolidin-2-yl}formamido)-5-carbamimidamido-N-(carbamoylmethyl)pentanamide
2-({1-[13-benzyl-10-(2-carbamoylethyl)-7-(carbamoylmethyl)-16-[(4-methoxyphenyl)methyl]-20,20-dimethyl-6,9,12,15,18-pentaoxo-1,2-dithia-5,8,11,14,17-pentaazacycloicosane-4-carbonyl]pyrrolidin-2-yl}formamido)-5-carbamimidamido-N-(carbamoylmethyl)pentanamide
2-({1-[19-benzyl-16-(2-carbamoylethyl)-13-(carbamoylmethyl)-22-[(4-methoxyphenyl)methyl]-12,15,18,21,24-pentaoxo-7,8-dithia-11,14,17,20,23-pentaazaspiro[5.19]pentacosane-10-carbonyl]pyrrolidin-2-yl}formamido)-5-carbamimidamido-N-(carbamoylmethyl)pentanamide
(4S,7R,10R,13S,16R,19S,22S,25S,28R,31R,34R,37R)-19,34-bis(4-aminobutyl)-37-{2-[(2R)-2-aminopropanamido]acetamido}-13,25,28-tribenzyl-31-(carbamoylmethyl)-10,16-bis[(1R)-1-hydroxyethyl]-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecaazacyclooctatriacontane-4-carboxylic acid
19,34-bis(4-aminobutyl)-37-[2-(2-aminopropanamido)acetamido]-25,28-dibenzyl-31-(carbamoylmethyl)-10,16-bis(1-hydroxyethyl)-7-(hydroxymethyl)-13-[(4-hydroxyphenyl)methyl]-22-(1H-indol-2-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecaazacyclooctatriacontane-4-carboxylic acid
37-{2-[2-(6-amino-2-{2-[2-(2-{[1-(2-{2-[2-({1-[2-(2-{2-[2-(2-amino-3-hydroxypropanamido)propanamido]-3-carbamoylpropanamido}-3-hydroxypropanamido)-3-carbamoylpropanoyl]pyrrolidin-2-yl}formamido)propanamido]-4-(methylsulfanyl)butanamido}propanoyl)pyrrolidin-2-yl]formamido}-5-carbamimidamidopentanamido)-4-carboxybutanamido]-5-carbamimidamidopentanamido}hexanamido)propanamido]acetamido}-19,34-bis(4-aminobutyl)-13,25,28-tribenzyl-31-(carbamoylmethyl)-10,16-bis(1-hydroxyethyl)-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecaazacyclooctatriacontane-4-carboxylic acid
37-[2-(2-{6-amino-2-[2-(2-{2-[(1-{2-[2-(2-{[1-(2-{2-[2-(2-{2-[2-amino-3-(4-hydroxyphenyl)propanamido]-3-hydroxypropanamido}propanamido)-3-carbamoylpropanamido]-3-hydroxypropanamido}-3-carbamoylpropanoyl)pyrrolidin-2-yl]formamido}propanamido)-4-(methylsulfanyl)butanamido]propanoyl}pyrrolidin-2-yl)formamido]-5-carbamimidamidopentanamido}-4-carboxybutanamido)-5-carbamimidamidopentanamido]hexanamido}propanamido)acetamido]-19,34-bis(4-aminobutyl)-13,25,28-tribenzyl-31-(carbamoylmethyl)-10,16-bis(1-hydroxyethyl)-7-(hydroxymethyl)-22-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecaazacyclooctatriacontane-4-carboxylic acid
6-(4-aminobutyl)-12-benzyl-3-[1-(benzyloxy)ethyl]-9-(1H-indol-3-ylmethyl)-1,4,7,10,13-pentaazacycloicosane-2,5,8,11,14-pentone
2-{[1-(6-amino-2-{[1-(2-amino-5-carbamimidamidopentanoyl)pyrrolidin-2-yl]formamido}hexanoyl)pyrrolidin-2-yl]formamido}-N-[3-carbamoyl-1-({1-[(1-{[({1-[(1-carbamoylpentyl)carbamoyl]-3-methylbutyl}carbamoyl)methyl]carbamoyl}-2-phenylethyl)carbamoyl]-2-phenylethyl}carbamoyl)propyl]pentanediamide
2-{[1-(6-amino-2-{[1-(2-amino-5-carbamimidamidopentanoyl)pyrrolidin-2-yl]formamido}hexanoyl)pyrrolidin-2-yl]formamido}-N-{3-carbamoyl-1-[(1-{[1-({[(1-{[1-carbamoyl-3-(methylsulfanyl)propyl]carbamoyl}-3-methylbutyl)carbamoyl]methyl}(methyl)carbamoyl)-2-phenylethyl]carbamoyl}-2-phenylethyl)carbamoyl]propyl}pentanediamide
2-{[1-(6-amino-2-{[1-(2-amino-5-carbamimidamidopentanoyl)pyrrolidin-2-yl]formamido}hexanoyl)pyrrolidin-2-yl]formamido}-N-{3-carbamoyl-1-[(1-{[1-({1-[(1-{[1-carbamoyl-3-(methylsulfanyl)propyl]carbamoyl}-3-methylbutyl)carbamoyl]-2-(1H-indol-3-yl)ethyl}carbamoyl)-2-phenylethyl]carbamoyl}-2-(1H-indol-3-yl)ethyl)carbamoyl]propyl}pentanediamide
2-{[1-(6-amino-2-{[1-(2-amino-5-carbamimidamidopentanoyl)pyrrolidin-2-yl]formamido}hexanoyl)pyrrolidin-2-yl]formamido}-N-{3-carbamoyl-1-[(1-{[1-({1-[(1-{[1-carbamoyl-3-(methylsulfanyl)propyl]carbamoyl}-3-methylbutyl)carbamoyl]-2-(1H-indol-3-yl)ethyl}carbamoyl)-2-phenylethyl]carbamoyl}-2-phenylethyl)carbamoyl]propyl}pentanediamide
2-{[1-(6-amino-2-{[1-(2-amino-5-carbamimidamidopentanoyl)pyrrolidin-2-yl]formamido}hexanoyl)pyrrolidin-2-yl]formamido}-N-[3-carbamoyl-1-({1-[(1-{[1-({1-[(1-carbamoyl-3-methylbutyl)carbamoyl]-3-methylbutyl}carbamoyl)-2-(1H-indol-3-yl)ethyl]carbamoyl}-2-phenylethyl)carbamoyl]-2-(1H-indol-3-yl)ethyl}carbamoyl)propyl]pentanediamide
1-(6-amino-2-{[1-(2-amino-5-carbamimidamidopentanoyl)pyrrolidin-2-yl]formamido}hexanoyl)pyrrolidine-2-carboxylic acid
2-{2-[2-(2-amino-3-phenylpropanamido)-3-phenylpropanamido]acetamido}-N-[1-carbamoyl-3-(methylsulfanyl)propyl]-4-methylpentanamide
2-(3-carboxy-2-acetamidopropanamido)pentanedioic acid
2-{2-[2-(2-aminopropanamido)-4-methylpentanamido]propanamido}-4-methylpentanoic acid
(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-aminopropanamido]-3-hydroxypropanamido]-3-hydroxybutanamido]-3-hydroxybutanamido]-3-hydroxybutanamido]-N-[(1S)-1-{[(1S)-1-carbamoyl-2-hydroxypropyl]carbamoyl}-2-(4-hydroxyphenyl)ethyl]butanediamide
2-[3-(1H-imidazol-4-yl)-2-[(5-oxopyrrolidin-2-yl)formamido]propanamido]acetic acid
6-amino-2-[2-(2-amino-3-hydroxybutanamido)-3-hydroxypropanamido]hexanoic acid
4-(2-{2-[2-(2-amino-5-carbamimidamidopentanamido)-5-carbamimidamidopentanamido]-4-methylpentanamido}-3-methylpentanamido)-4-({1-[(1-{[1-({1-[(1-{[1-({4-carbamimidamido-1-[(carboxymethyl)carbamoyl]butyl}carbamoyl)ethyl]carbamoyl}ethyl)carbamoyl]-2-(4-hydroxyphenyl)ethyl}carbamoyl)-3-carboxypropyl]carbamoyl}ethyl)carbamoyl]-2-carboxyethyl}carbamoyl)butanoic acid
4-(2-{2-[2-(2-amino-5-carbamimidamidopentanamido)-5-carbamimidamidopentanamido]-4-methylpentanamido}-3-methylpentanamido)-4-({1-[(1-{[1-({1-[(1-{[1-({4-carbamimidamido-1-[(carboxymethyl)carbamoyl]butyl}carbamoyl)ethyl]carbamoyl}-2-hydroxypropyl)carbamoyl]-2-(4-hydroxyphenyl)ethyl}carbamoyl)-3-carboxypropyl]carbamoyl}-2-carbamoylethyl)carbamoyl]-2-carboxyethyl}carbamoyl)butanoic acid
1-{2-[2-(2-{6-amino-2-[2-(2-amino-5-carbamimidamidopentanamido)-5-carbamimidamidopentanamido]hexanamido}propanamido)-3-hydroxypropanamido]acetyl}pyrrolidine-2-carboxylic acid
2-[2-(2-amino-5-carbamimidamidopentanamido)acetamido]butanedioic acid
3-[2-(2-amino-5-carbamimidamidopentanamido)acetamido]-3-[(1-carboxy-2-hydroxyethyl)carbamoyl]propanoic acid
3-[2-(2-amino-5-carbamimidamidopentanamido)-3-phenylpropanamido]-3-[(1-carboxy-2-hydroxyethyl)carbamoyl]propanoic acid
2-[(1-{2-[2-(2-amino-3-carboxypropanamido)-3-hydroxypropanamido]-3-carboxypropanoyl}pyrrolidin-2-yl)formamido]-5-carbamimidamidopentanoic acid