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N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2-(trifluoromethyl)benzamide
4-methoxy-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-4-(prop-2-en-1-yl)piperidine
N-(3-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}phenyl)pyridine-4-carboxamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[4-(propan-2-yl)piperidin-1-yl]methyl}piperidin-2-one
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-(3-phenylpropyl)-1,4-diazepan-2-one
1-(4-{2,8-diazaspiro[4.5]decane-2-sulfonyl}phenyl)-3-methylurea
2-{2-methyl-6-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyrimidin-4-yl}ethan-1-amine
3-fluoro-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}pyridine-4-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-4-(2-oxopyrrolidin-1-yl)butanamide
2-{8-[1-(4-methylphenyl)cyclopropanecarbonyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
5-(morpholin-4-ylmethyl)-N-(2-phenylpropyl)-1,2-oxazole-3-carboxamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-3-(1H-imidazol-1-ylmethyl)piperidine
(1S,6R)-3-{[2-(difluoromethoxy)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
(3S,4S)-4-cyclopropyl-1-(pyrimidin-5-ylmethyl)pyrrolidine-3-carboxylic acid
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
4-methoxy-3-{2-oxa-7-azaspiro[4.5]decane-7-carbonyl}benzene-1-sulfonamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N,6-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-cyclopentyl-8-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(4-fluorophenyl)ethyl]-1,3-oxazole-4-carboxamide
4-[(2-methylphenyl)sulfanyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
1-methyl-3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazole
5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-2-methoxypyridine
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N,N-bis(prop-2-en-1-yl)acetamide
(1R,5S)-N-{4-chloro-3-[(propan-2-yl)carbamoyl]phenyl}-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3R,4R)-1-[1-(2-fluorophenyl)piperidin-4-yl]-3,4-dimethylpyrrolidin-3-ol
methyl 3-cyclobutaneamido-5-[(2,2-dimethylpropyl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decane
6-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)-1H-indole
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(2-hydroxyethyl)phenyl]-3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
3-(2,5-dichlorophenyl)-2,5-dimethylpyrazine
3-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-ol
5-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
(4aR,7aS)-1-(2-methoxyethyl)-4-[(3E)-pent-3-enoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-(quinolin-8-yl)urea
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(2-phenylethyl)-1H-1,2,3-triazole
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-cyclopropylacetamide
2-(pyridin-3-yl)-5-[4-(thiophen-3-ylmethyl)piperazine-1-carbonyl]pyrimidine
5-{4-hydroxy-1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
8-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-(2-chlorophenyl)-3-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
3-[1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-2-yl]pyridine
2-{4-[(2,3-difluorophenyl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one