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N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,3-thiazole-5-carboxamide
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-[2-(dimethylamino)ethyl]-4-[4-(furan-2-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
4-benzyl-3-ethyl-1-(4-methylpyrimidine-5-carbonyl)-1,4-diazepan-5-one
2-methoxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyridine-4-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(furan-3-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
8-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
6-(difluoromethyl)-2-[3-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N-(1H-indol-6-ylmethyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(6-phenoxypyridin-3-yl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
N-(3-methoxyphenyl)-1-(2-{[(1-methyl-1H-pyrrol-2-yl)methyl]amino}ethyl)-1H-1,2,3-triazole-4-carboxamide
({3-methyl-1-[2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)(pyridin-2-ylmethyl)amine
3-{2-[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
N-{[5-(quinolin-6-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
1-(2-fluorophenyl)-4-[(4-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
5-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-methoxy-2-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
N-[(3-chlorophenyl)methyl]-3-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]propanamide
2-(2-hydroxyethyl)-9-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amino}-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
(3aR,6aR)-2-(2-chloro-4-fluorobenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-hydroxy-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-{5-[1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(morpholin-2-ylmethyl)acetamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
N-(2-hydroxyethyl)-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
6-(4-butylpiperazin-1-yl)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
1-[4-(hydroxymethyl)pyridine-2-carbonyl]-4-(propan-2-yl)-1,4-diazepan-6-ol
1-(azepan-1-yl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
[3-(cyclopropylmethyl)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]methanol
3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-4-(2-phenylethyl)piperazin-2-one
methyl (2S,4S)-1-[(2-ethoxyphenyl)methyl]-4-(4-methylbenzamido)pyrrolidine-2-carboxylate
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-N-[(2,3,4-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
ethyl 3-{[2-(4-methoxyphenyl)phenyl]carbamoyl}piperidine-1-carboxylate
1-methyl-4-{2-[4-(2-methylpropyl)phenyl]pyridine-4-carbonyl}piperazine
N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-6-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
[(8-chloroquinolin-2-yl)methyl](methyl)[2-(pyridin-2-yl)ethyl]amine
(2S)-2-{[5-(3-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}-3-methylbutanamide
3-acetyl-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-(1,2-oxazol-3-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-[2-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-4-(pyridin-3-yl)phenoxy]acetic acid
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-(2-methylbutan-2-yl)pyridine-3-carbonitrile
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(3-fluorophenyl)methyl](2-methoxyethyl)amine
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,3-diol
4-(5-methylpyridin-2-yl)-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-ol