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4-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyridine
8-[1-(methylsulfanyl)propan-2-yl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-({1-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
N-(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
3-[(4-benzyl-2-oxopyrrolidin-1-yl)methyl]-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide
1-(2-fluorophenyl)-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazine
N-[(3-fluoro-4-methoxyphenyl)methyl]-1-methylpiperidine-2-carboxamide
4-[5-({8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
6-methoxy-3-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1,2-dihydroquinolin-2-one
3-{4-oxo-4-[2-(pyridin-2-yl)pyrrolidin-1-yl]butyl}-3,4-dihydroquinazolin-4-one
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-[(3,4-dimethoxyphenyl)methyl]-3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidine
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
2-(2-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-(2,3-dihydro-1H-inden-4-yl)-3-(thiophene-2-carbonyl)piperidine-1-carboxamide
N,N-dimethyl-5-[(2-oxo-1,2-dihydroquinoxalin-1-yl)methyl]furan-2-carboxamide
2-(5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-(methylsulfanyl)-N-[(5-oxo-1-phenylpyrrolidin-3-yl)methyl]-1,3-thiazole-4-carboxamide
3-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-7-fluoro-1,2-dihydroquinolin-2-one
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
(4aS,7aR)-1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-6-ethylpyrimidin-4-amine
2-{4-[3-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}-1,3-benzoxazole
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
6-methyl-N4-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)pyrimidine-2,4-diamine
1-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}phenyl)-1H-1,2,4-triazole
6-(2-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1,4-dithiepan-6-amine
(2S,4S)-4-[4-({[(3-cyanophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}benzamide
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-fluoro-2-methylphenyl)acetamide
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,3-diol
1-propanoyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
6-[2,6-dimethyl-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
N-(adamantan-2-ylmethyl)-6-[(2-ethylpiperidin-1-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(3,5-dimethoxyphenyl)-3-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
2-[1-(1-methanesulfonylpyrrolidine-2-carbonyl)azetidin-3-yl]pyridine
1-{2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyrrolidin-2-one
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
(4aS,7aR)-1-hexanoyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(5-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}-1H-1,3-benzodiazol-2-yl)methanol