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3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
1-(2-oxo-2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,2-dihydropyrimidin-2-one
2-(4-chlorobenzoyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aS)-2-(ethanesulfonyl)-5-[2-(2-fluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
(2S)-2-amino-4-(methylsulfanyl)-1-[2-(morpholin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]butan-1-one
N-({7-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
(2S,4R)-1-acetyl-N-ethyl-4-[3-(trimethyl-1H-pyrazol-4-yl)propanamido]pyrrolidine-2-carboxamide
(3R,4R)-1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-ethylpiperazin-1-yl)ethan-1-one
4-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]-1-ethyl-N,N-dimethylpiperidin-4-amine
(3S,4S)-4-(dimethylamino)-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
N,N-diethyl-4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-8-{[4-(5-methylfuran-2-yl)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3S,4S)-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
1-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidine-4-carboxylic acid
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-amine
1-[(3-fluoro-2-methylphenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-cycloheptyl-5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]piperidin-2-one
5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-[2-(cyclohexylmethyl)morpholine-4-carbonyl]pyridin-2-ol
7-(morpholin-4-ylmethyl)-4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(3S)-1-benzylpiperidin-3-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
5-propyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(3-{4-[(5-hydroxyadamantan-2-yl)amino]piperidin-1-yl}phenyl)-2-methoxybenzamide
1-(6-hydroxy-4-{[3-(3-methoxyphenyl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
1-(pyridin-2-ylmethyl)-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
4-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-{1-[4-(quinolin-5-yloxy)piperidine-4-carbonyl]pyrrolidin-3-yl}acetamide
4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(1,2,4-thiadiazol-5-yl)benzamide
5-acetyl-N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
2-ethoxy-4-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
2-{1-[(2-methylphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,2,5-thiadiazole-3-carboxamide
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-methylbut-2-en-1-yl)piperidin-3-yl]methanol
4-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}pyridine-4-carbonyl)morpholine
3-amino-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
2-[4-(methylsulfanyl)phenyl]-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-imidazole
4-(5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)-1H-pyrazole
9-(6-methylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[2-(4-methoxyphenyl)ethyl][(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl][(1-methylpiperidin-4-yl)methyl]amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(4H-1,2,4-triazol-4-yl)benzamide
2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid