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2-({[(5-carboxyfuran-2-yl)methyl]carbamoyl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
3-(1H-imidazol-2-yl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
6-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]pyridine-2-carboxamide
[(3R,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-ol
2-tert-butyl-5-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]pyrimidin-4-ol
3-[(2-hydroxyethyl)({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
1-[benzyl(methyl)amino]-3-[4-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-(2-chlorophenyl)-5-cyclobutyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
2-methyl-1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)propan-1-one
1'-(2-methyl-1,3-thiazole-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-ethyl-1-[4-(2-fluorophenoxy)phenyl]-3-[2-(morpholin-4-yl)ethyl]urea
2-(4-{[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
2-(2-methoxyphenoxy)-N-{[1-(pyrimidin-5-ylmethyl)piperidin-3-yl]methyl}acetamide
ethyl 4-[(2-hydroxy-5-phenylphenyl)methyl]piperazine-1-carboxylate
3-[3-(2-methoxyphenoxy)azetidin-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
N-(2-acetamidophenyl)-2-[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amino]acetamide
9-(3-phenoxypropanoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1H-indol-3-yl)-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}acetamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
8-(6-ethyl-2-methylpyrimidin-4-yl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-[(3-methoxyphenyl)methyl]-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(morpholin-4-yl)-2-oxoethyl]-1,4-diazepane-6-carboxylic acid
1-[1'-(quinolin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-ethyl-4-(1H-imidazol-2-ylmethyl)-1-(propan-2-yl)piperazine
(2S)-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-4-(propan-2-yl)pyrimidin-2-amine
5-amino-N-[(3S,5S)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
N-(2,6-difluorophenyl)-2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
(1R,2S)-2-[(5-fluoroquinazolin-4-yl)amino]cyclopentane-1-carboxamide
(5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}furan-2-yl)methanol
3-methyl-N-{[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]methyl}but-2-enamide
5-[(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-cyclopropyl-1H-1,2,4-triazole
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,4-dimethyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
8-(6-methylpyridine-2-carbonyl)-1-oxa-8-azaspiro[4.5]decane
8-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-ethyl-3-{2-oxo-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
1-[4-(1-butyl-1H-1,2,4-triazol-5-yl)-1,3-thiazol-2-yl]-4-phenylpiperazine
[1-(1-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanamine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
N-ethyl-1-(5-ethylpyrimidin-2-yl)pyrrolidine-3-carboxamide
[1-(1-phenylmethanesulfonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
2-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)phenol
2-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[3-(1H-imidazol-1-yl)propyl]-9-(9H-purin-6-yl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,3R)-N1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]cyclopentane-1,3-diamine
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-[methyl(1-methylpiperidin-4-yl)amino]ethan-1-one
6-[2-(pyridin-3-yl)-1H-imidazol-1-yl]-1H-indole