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methyl 4-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}methyl)-1H-pyrazole-3-carboxylate
2-(pentan-2-yl)-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazole
2-methyl-1-(2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1H-indole-3-carbonitrile
(2-{[4-(2,3-difluoro-4-methylbenzoyl)piperazin-1-yl]methyl}phenyl)methanol
8-methoxy-2-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}quinoline
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
N-(4-methoxy-2-methylphenyl)-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}propanamide
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
5,7-dimethyl-3-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrazolo[1,5-a]pyrimidine
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2-methoxy-5-methylphenyl)acetic acid
(3R,4S)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4-(3-methoxyphenyl)pyrrolidin-3-amine
3-({[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}methyl)-N,N-dimethylbenzamide
1-ethyl-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
N-{2-methoxy-4-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamido]phenyl}butanamide
1-methyl-4-[(4-methyl-5-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]piperazine
N-[2-(3-fluorophenyl)ethyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)benzonitrile
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
methyl 3-(furan-2-amido)-6-(piperidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
4-{4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazin-1-yl}benzonitrile
2,5-dimethyl-3-(4-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
5-({2-[ethyl(3-methylphenyl)amino]ethyl}carbamoyl)-1H-imidazole-4-carboxylic acid
N-(2-fluoro-4-methylphenyl)-2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)propanamide
N-[4-(2-benzyl-3-oxopiperazine-1-carbonyl)phenyl]-2-(dimethylamino)acetamide
1-(2-fluoro-6-methoxybenzoyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-cyclopropyl-N-[2-(2,3-dimethoxyphenyl)ethyl]pyrimidine-5-carboxamide
(1S,3R)-3-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopentane-1-carboxamide
N-{2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]ethyl}-N-methylmethanesulfonamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(dimethyl-1,3-oxazole-5-carbonyl)piperidine-4-carboxylic acid
9-[(4-acetylphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1-benzothiophen-3-yl)-N-methylbenzamide
N-{1-[(2-chloro-5-ethoxy-4-propoxyphenyl)methyl]piperidin-4-yl}acetamide
4-{[(dimethyl-1,3-thiazol-5-yl)methyl](methyl)amino}-2-methylbutan-2-ol
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-4-carboxamide
3-{4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-1-yl}-1,2-benzothiazole
2,7-bis[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-({1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]piperidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
(4aR,7aS)-1-methyl-4-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(carbamoylmethoxy)-N-(2-hydroxy-3-phenylpropyl)benzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
3-(2,3-dihydroxypropyl)-1-[2-fluoro-3-(trifluoromethyl)phenyl]-3-methylurea
N-(5-ethyl-1,3,4-oxadiazol-2-yl)-1-(morpholine-4-carbonyl)piperidin-4-amine
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1,3-dimethyl 5-[(4-cyanopiperidine-1-carbonyl)amino]benzene-1,3-dicarboxylate
5-({[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}methyl)-1-methylpyrrolidin-2-one
N-[(3R,4R)-3-hydroxy-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl]pyrazine-2-carboxamide
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})methylamine