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4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N,N-bis(prop-2-en-1-yl)benzamide
2-{[2-amino-6-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)pyrimidin-4-yl]amino}ethan-1-ol
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(2-hydroxyethyl)-N-methylbenzamide
1-methyl-N-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
5-[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-2-yl]-N-(1H-pyrazol-3-yl)thiophene-2-carboxamide
4-[1-(1-{[3-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)ethyl]morpholine
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2H-1,2,3-benzotriazol-2-yl)ethan-1-one
N-cyclopentyl-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-(2-chlorophenyl)-3-methyl-N-[3-(methylsulfanyl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(3,4-difluorophenyl)-1-[2-(morpholin-4-yl)benzoyl]piperidin-3-amine
1-{[3-ethoxy-4-(5-fluoro-2-methylphenoxy)phenyl]methyl}pyrrolidine
3-{[(furan-3-ylmethyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
4-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(methoxymethyl)cyclopentyl]benzamide
N-methyl-3-phenyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
2-methyl-7-(3-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
3-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)propanamide
N-{2-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide
1-benzyl-4-[(2,6-difluorophenyl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
6-(4-methoxyphenyl)-9-[2-(pyridin-2-ylsulfanyl)acetyl]-6,9-diazaspiro[4.5]decan-7-one
1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(3-methyl-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(2S)-2-acetamido-3-(1H-imidazol-4-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-chloro-N-({1-[2-(1H-imidazol-4-yl)acetyl]piperidin-3-yl}methyl)benzamide
N-methyl-N-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidin-2-amine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-1-[2-hydroxy-2-(thiophen-2-yl)ethyl]urea
5-(1H-indole-5-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
ethyl 2-[({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)(methyl)amino]acetate
2-phenyl-N-(pyridin-3-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-chloro-5-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-N-methylbenzamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-ol
2-(dimethyl-1,3-thiazol-5-yl)-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)acetamide
3-[(4-methoxyphenyl)methyl]-5-methyl-1-propyl-1H-1,2,4-triazole
N-[2-(4-hydroxy-3-methoxyphenyl)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-{2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-oxoethyl}piperazin-2-one
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(pyridin-4-ylmethyl)amine
4-[(dimethylamino)methyl]-1-(3-fluoro-4-methylbenzenesulfonyl)azepan-4-ol
4-ethyl-3-{1-[5-(methanesulfonylmethyl)pyridin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-1-(5-methoxyfuran-2-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-{[(4-methyl-1,3-thiazol-2-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
(4aR,7aS)-1-(2-methylpropyl)-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-benzyl-3-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[4-(3-methylphenyl)phenyl]-1-[(2-oxo-1,3-oxazolidin-5-yl)methyl]piperidine-4-carboxamide
1-[(4-fluorophenyl)methyl]-4-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperazin-2-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-4-hydroxy-2-(pyridin-4-yl)pyrimidine-5-carboxamide