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1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(1S,4S)-5-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-({[(3R,4R)-1-(3,5-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
2-chloro-N-[2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]benzamide
ethyl 4-{[5-(2,5-dimethoxyphenyl)-2-hydroxyphenyl]methyl}piperazine-1-carboxylate
4,4-difluoro-1-[(2-methoxy-3,5-dimethylphenyl)methyl]piperidine
3-cyclopropyl-1-[2-fluoro-5-(trifluoromethyl)phenyl]-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(pyrrolidin-3-yl)benzamide
3-[(1-acetylpiperidin-4-yl)oxy]-N-(2,3-dihydro-1H-inden-1-yl)-4-methoxybenzamide
N-[4-(3-methylphenyl)phenyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-4-carboxamide
1-(3-cyano-4-methylphenyl)-3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}urea
2-(6-aminopyridin-3-yl)-2-{methyl[(3-methyl-1H-indol-2-yl)methyl]amino}acetic acid
1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
3,6-dimethyl-N-[3-(pyridin-3-yloxy)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-{3-oxo-3-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]propyl}imidazolidine-2,4-dione
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(5-fluoropyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
1-(2,3-dimethylphenyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
8-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(5-{3-[(4-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)phenol
3,3-diethyl-1-[4-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)phenyl]urea
N-methyl-N-[2-(oxan-2-yl)ethyl]-4-(piperidin-1-yl)benzamide
1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
1-(3-methylpyridin-2-yl)-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperazine
1-(3-methoxypropanoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-(furan-3-ylmethyl)-4-(piperidine-1-sulfonyl)-1,4-diazepane
(1S,5R)-6-benzyl-3-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2H-1,3-benzodioxol-5-ylmethyl)(methyl){[(1R,5S,6R)-3-(morpholine-4-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}amine
2-methyl-5-[2-(3-phenoxypropyl)phenyl]-1,3,4-oxadiazole
(3S,6S)-6-benzyl-3-methyl-4-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-(methoxymethyl)-5-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyrimidine
1-ethyl-N-methyl-3-(thiomorpholine-4-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
8-[2-(methylsulfanyl)propanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-cyano-N-({1-[(4,5-dimethylfuran-2-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
(3S)-3-[({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)amino]azepan-2-one
6-[2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyrimidin-4-ol
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
N-methyl-6-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-cyclopropanecarbonyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[(2-{[1-(thiophen-2-yl)butyl]carbamoyl}phenyl)amino]acetic acid
N,5-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
4-[4-(2-chloro-6-methoxyphenyl)phenyl]piperidin-4-ol
2-methyl-4-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]pyrimidine
N-[1-(4-methanesulfonylphenyl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylthian-4-amine