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(3aS,7aR)-5-methyl-2-[6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carbonyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-(1,4-dioxan-2-ylmethyl)-7-fluoro-3,4-dihydroquinazolin-4-one
3-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-benzyl-4-[4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperazin-2-one
6-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-ethyl-N-methylpyridine-3-carboxamide
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-(3-methoxypropyl)-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
3-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
2-[1-(3-methylbutyl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
1-(3-methoxyphenyl)-5-methyl-4-[3-(1H-pyrrol-1-yl)propanoyl]piperazin-2-one
N-ethyl-5-{[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-4-methyl-N-(pyridin-3-ylmethyl)benzamide
2-methyl-5-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]-3,4-dihydropyrimidin-4-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-methyl-4-phenylpyrimidine-5-carboxamide
methyl(oxolan-2-ylmethyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-[(4-chloro-1,3-dimethyl-1H-pyrazol-5-yl)formamido]-N-methylpentanamide
N,N,4-trimethyl-6-{[1-(4-methyl-1,4-diazepan-1-yl)hex-5-en-2-yl]oxy}pyrimidin-2-amine
2-[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carboxylic acid
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(4-methylmorpholin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
{3-[(2-methylphenyl)methyl]-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}methanol
8-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-ethyl-5-methyl-N-(pyridin-4-ylmethyl)-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
5,6-dimethyl-3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyridine-3-carboxamide
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carbonyl}piperidine
1-[4-(benzyloxy)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-(4-ethylpiperazin-1-yl)-3-(3-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
9-ethyl-4-(4-ethyl-5-methylthiophene-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
4-[4-(thian-4-yl)piperazin-1-yl]pyrimidine
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-N-cyclobutylbenzene-1-sulfonamide
2-(5-methyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
(4aS,8aS)-2-(1,3-thiazol-4-ylmethyl)-decahydroisoquinolin-4a-ol
(2E)-N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
3-[(4aR,7aS)-4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(1-benzofuran-2-ylmethyl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
3-[(2-oxopyrrolidin-1-yl)methyl]-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
4-[(2,4-dimethoxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methoxy-5-[3-(4-methylpiperazin-1-yl)pyrrolidine-1-carbonyl]phenol
1-methyl-2-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
7-chloro-2-{[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[2-(5-methylfuran-2-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(3S)-3-ethyl-4-({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)morpholine
methyl(thiophen-2-ylmethyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-cyclohexyl-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methylbenzamide
6-methyl-5-{5-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine