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(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
methyl 2-(5-{1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
(1R,5R)-3-(3-fluoropyridine-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
4-(4,4-difluoropiperidine-1-carbonyl)-2,6-dimethylpyridine
N-(3-fluorophenyl)-6-[3-(1H-indol-3-yl)propanoyl]-6-azaspiro[2.5]octane-1-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-(quinolin-2-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
6-[(diethylamino)methyl]-N-[2-(morpholin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1R,2R)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-2-phenylcyclopropane-1-carboxamide
methyl 4-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)butanoate
6-(5-methoxypyrimidin-2-yl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-oxoazepan-1-yl)propanamide
2-methoxy-1-{4-[4-(3-propoxypiperidine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
3-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
(4aR,8aR)-7-[2-(benzenesulfonyl)ethyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
3-[(cyclohex-1-en-1-ylmethyl)sulfamoyl]-N-(2-methoxyethyl)benzamide
5-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-3-phenyl-1,2-oxazole
(5S)-5-(4-{[4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrrolidin-2-one
1-(4-hydroxy-4-phenylpiperidin-1-yl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
(3S,4R)-1-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
1-(4-fluorophenyl)-4-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]piperazine
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
4-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
2-[2-(azocan-1-yl)acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethane-1-sulfonamide
1-ethyl-5-{[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-({1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
(5R)-5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
1-{1-[5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}-3-phenylpropan-1-one
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-[(3R)-pyrrolidin-3-yl]urea
1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)ethan-1-one
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-(3-methylphenyl)propanamide
(4aR,7aS)-1-benzyl-4-[(2,6-dimethylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(4-methylpyridin-2-yl)propyl]-1H-pyrazole-3-carboxamide
4-{5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2,4-oxadiazol-3-yl}-1H-indole
4-[4-(benzyloxy)butyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-[(propylamino)methyl]piperidin-2-one
N-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
6-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}thiomorpholine
2-(butan-2-yl)-1H-1,3-benzodiazole-5-carbonitrile
1-{4-[(2-cyclopentyl-2-phenylethyl)amino]piperidin-1-yl}ethan-1-one
4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-(propan-2-yl)-1H-pyrazole
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-[2-(pyridin-3-yloxy)ethyl]acetamide
9-[(2-fluoro-5-methylphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2,6-dimethyl-4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}quinoline
(3S,4S)-4-(naphthalen-2-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-3-ol
5-amino-4-chloro-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}oxy)pyrimidine
2-[4-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]acetamide