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2-(2,4-difluorophenoxy)-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
2-(2-chloro-6-fluorophenyl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-{[2,4-dimethyl-5-(1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazol-2-yl)phenyl]methyl}-1H-1,2,4-triazole
7-(cyclopropylmethyl)-2-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
2-(3-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}-1H-indol-1-yl)acetamide
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-methyl-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-{[3-(2-fluorophenyl)phenyl]methyl}-N-methyloxan-4-amine
5-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
3-ethyl-4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-[(3R,4S)-4-cyclopropyl-1-(3-methoxypropyl)pyrrolidin-3-yl]-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
1-[(5-chlorothiophen-2-yl)methyl]-3-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)urea
N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)-N-(quinolin-6-ylmethyl)benzamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-N-(pyridin-3-yl)propanamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{3-[(4-fluorophenyl)methoxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(1-benzothiophen-5-ylmethyl)-4-hydroxybenzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-methanesulfonamido-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-5-(propan-2-yl)-1,2-oxazole
3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
3-[4-(9H-fluoren-2-ylmethyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
N-methyl-5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)azepan-4-amine
N-{1-[(4-methylpiperidin-1-yl)sulfonyl]azepan-3-yl}pyrrolidine-1-carboxamide
N-(2-chlorophenyl)-3-[1-(oxolan-2-ylmethyl)piperidin-4-yl]propanamide
5-[(2R,6R)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1H-1,3-benzodiazole
N-[2-(dimethylamino)ethyl]-N-{[7-fluoro-2-(2-methylphenyl)quinolin-3-yl]methyl}-4-methylbenzamide
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
N,1-dimethyl-2-(morpholin-4-yl)-N-[1-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-{1-[2-(1H-pyrazol-1-yl)acetyl]pyrrolidin-2-yl}-N-(1,2,3-thiadiazol-5-yl)thiophene-2-carboxamide
8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{3-[3-(benzyloxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-cyclopropyl-1-(2,4-dichlorophenyl)-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazole
4-{4-[2-(1H-imidazol-2-yl)phenoxy]butyl}morpholine
N-(3-hydroxy-3-phenylpropyl)-N-methyl-4-propylpyrimidine-5-carboxamide
2-benzyl-8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-ethyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(2,2,2-trifluoroethyl)acetamide
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-{1-[(5-ethylfuran-2-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-(2,3-dihydro-1H-indene-5-carbonyl)-3-(1H-imidazol-2-yl)piperidine
5-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(2-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
1-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}benzoyl)piperidine
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl][(4-ethylphenyl)methyl]methylamine
2-chloro-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
1'-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]
11-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one