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2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
6-[({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-2-methylpyrimidin-4-ol
3-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-(2,6-dimethylpyridin-3-yl)urea
(1S,3R)-3-amino-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]cyclopentane-1-carboxamide
6-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-{[(3,4-difluorophenyl)carbamoyl]methyl}-3-methylbut-2-enamide
2-(1-benzothiophen-3-yl)-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetic acid
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-methylazepane-2-carboxamide
N-(cyclopropylmethyl)-3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-(2-methoxyethyl)benzamide
1-[(2-fluorophenyl)methyl]-4-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperazin-2-one
3-(3-methoxybenzoyl)-1-[(2,3,6-trifluorophenyl)methyl]piperidine
3-(aminomethyl)-4-(3-chloro-4-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-({[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}amino)-2-fluorobenzamide
[1-({[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}amino)cyclopentyl]methanol
[(2S,4R)-4-(dimethylamino)-1-[2-(pyridin-3-yl)quinoline-4-carbonyl]pyrrolidin-2-yl]methanol
2-[4-(2-phenoxyacetyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-2-phenylethane-1,2-dione
1-(3,5-dimethylphenyl)-4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}piperazin-2-one
N-ethyl-N'-(2-fluoro-5-methylphenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]butanediamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole
(4S)-4-acetamido-5-[(3S)-3-ethylmorpholin-4-yl]-5-oxopentanamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[2-(furan-2-yl)ethyl]pyridin-2-amine
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2-oxazol-3-amine
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
3-(piperidin-3-yl)-N-[4-(pyrrolidin-1-yl)butyl]benzamide
N-({1-[1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}methyl)acetamide
(1R,5R)-N,N-dimethyl-6-[3-(pyridin-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(1R,9S)-5-amino-12-cyclopentyl-3-(1,5-dimethyl-1H-pyrazol-4-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(3S,5R)-1-(1,3-benzothiazol-2-yl)-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
1-acetyl-N-butyl-N-[(3-methoxyphenyl)methyl]piperidine-4-carboxamide
5-ethyl-2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyrimidine
4-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidine-1-carbonyl)-2,3-dihydro-1H-imidazol-2-one
4-[1-benzyl-5-(2,3-dihydro-1H-inden-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
1-[(2-methoxyphenyl)methyl]-N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)(quinolin-5-ylmethyl)amine
N-cyclobutyl-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
N5-[(5-ethylpyridin-2-yl)methyl]-N6-(2-methoxyethyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-methyl-1-(2-methylphenyl)-4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
N3-[1-(4-fluorophenyl)-2-methylpropan-2-yl]piperidine-1,3-dicarboxamide
(3S,4S)-4-methoxy-N-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-(propan-2-yl)pyrrolidin-3-amine
3-[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(2,3-difluoro-6-methoxyphenyl)methyl]-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
(3R,4S)-3,4-dimethyl-1-(5-methyl-2-phenylfuran-3-carbonyl)piperidin-4-ol
ethyl 1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate