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3-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-N-(pyridin-3-yl)propanamide
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]pyridine-2-carbonyl}morpholine
2-(3-{[2-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
2-ethyl-4-methyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-5-carboxamide
1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
2-fluoro-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-5-sulfamoylbenzamide
5-(methoxymethyl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)furan-2-carboxamide
(3S)-1-benzyl-N-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-amine
({4-cyclopropyl-5-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(3aS,6aS)-5-[(2,3-difluoro-6-methoxyphenyl)methyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
(4aR,8aR)-7-(1-benzothiophen-2-ylmethyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
1-(4,6-dimethylpyridine-3-carbonyl)-4-(2-phenoxyethyl)piperazine
dimethyl(3-{2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-yl}piperidin-3-ol
4-(3-hydroxy-3-methylbutyl)-N-(oxan-4-yl)benzamide
2-amino-1-{6-methyl-5-[5-(6-methylpyridin-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
N-{2-[1-(2-{2-methyl-7-oxo-6H,7H-[1,3]oxazolo[5,4-d]pyrimidin-6-yl}acetyl)piperidin-4-yl]ethyl}acetamide
N-(2-methoxyethyl)-3,6-dimethyl-N-(thiophen-3-ylmethyl)-1-benzofuran-2-carboxamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(1,2-oxazol-3-ylmethyl)amine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
8-fluoro-2-({[(3R)-pyrrolidin-3-yl]amino}methyl)quinolin-4-ol
4-(4-phenylpiperazine-1-carbonyl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
3-(3-hydroxyquinoxalin-2-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylpropanamide
[(3R,4S)-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(3S,4S)-4-cyclopropyl-1-(1,5-dimethyl-1H-indole-2-carbonyl)pyrrolidine-3-carboxylic acid
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(5-methoxyfuran-2-carbonyl)piperidine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(3-methylbutyl)-2,3-dihydro-1H-indene-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-sulfamoylthiophene-2-carboxamide
(1-{5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperidin-4-yl)methanol
(2S)-2-[(5-fluoroquinazolin-4-yl)amino]-3-hydroxypropanamide
1-{5-[(cyclohexylamino)methyl]-2-methoxyphenoxy}-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[(2-methanesulfonylethyl)amino]methyl}piperidin-2-one
4-[2-(dimethylamino)acetyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
1-methyl-3-(2-methylpropyl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
N-[5-(4-acetyl-1,4-diazepane-1-carbonyl)-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazol-7-yl]acetamide
4-[(7-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1λ6-thiomorpholine-1,1-dione
3-[(2-aminopyrimidin-5-yl)methyl]-1-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-methylurea
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)amine
2-[3-fluoro-5-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{4-[({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]piperidin-1-yl}ethan-1-one
1-[benzyl(methyl)amino]-3-[4-({[2-(dimethylamino)ethyl]amino}methyl)phenoxy]propan-2-ol
9-(2-methoxyethyl)-1-methyl-4-[2-(pyridin-4-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
3-[(3,4-dimethylpiperazin-1-yl)methyl]-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
1-[(5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}thiophen-3-yl)methyl]pyrrolidine
1-[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]-3-(1H-indol-3-yl)propan-1-one
[(2-butyl-1H-imidazol-4-yl)methyl](methyl)[(3-phenyl-1H-pyrazol-5-yl)methyl]amine
1-(carbamoylmethyl)-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
N-{[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide