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(4aS,8aS)-2-[(2,6-difluorophenyl)methyl]-decahydroisoquinolin-4a-ol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
2-[(2S)-2-amino-2-cyclopropylacetyl]-N-(2-methoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridin-4-amine
N-(2-{[2-(pyridin-3-yl)pyrimidin-5-yl]formamido}ethyl)pyridine-3-carboxamide
7-cyclopentyl-2-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-(3-methoxyphenyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-pyrazole-4-carboxamide
2-(dimethyl-1,3-thiazol-4-yl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
(2S)-1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-methyl-2-phenylpiperazine
1-[(3,5-dimethylphenyl)methyl]-4-[(5-hydroxy-2-methoxyphenyl)methyl]piperazin-2-one
1-[2-(pyridin-3-yl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
4-{2-[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}morpholine
4-(2,3-difluorobenzoyl)-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(3,4,5-trimethoxyphenyl)pyridin-2-amine
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-amine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
2-(1,3-thiazol-4-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
5-[(adamantan-1-ylmethyl)(methyl)amino]-1-[(4-methoxyphenyl)methyl]azepan-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-hydroxy-N-methylpyrazine-2-carboxamide
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
3-propyl-4-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}morpholine
(1S,6R)-3-methyl-9-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
9-[(4-methoxyphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
8-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
methyl 2-(azepane-1-sulfonyl)-6-(3-methoxybenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
3-(1,4-oxazepane-4-sulfonyl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
2-amino-6-benzoyl-4-(4-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
2-{[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amino]methyl}benzonitrile
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-benzyl-N-methyl-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-amine
7-fluoro-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
4-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}-2-ethylpyrimidine
1-(azepan-1-yl)-4-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}butane-1,4-dione
2-benzyl-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)morpholine
1-(3-methoxybenzoyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazine
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-{[3-(pyrrolidin-1-yl)phenyl]methyl}urea
N-(1-methoxypropan-2-yl)-1-{2-[(prop-2-en-1-yl)amino]benzoyl}piperidine-4-carboxamide
3-(4-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(4-methylphenyl)methyl]piperidin-4-ol