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methyl 1-{2-hydroxy-3-[3-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
2-(2-methylpropyl)-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
3-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
6-ethoxy-2-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}quinoline
N-cyclopropyl-3-(2-methylpropyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
N-ethyl-N-{[1-(1H-imidazol-4-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}furan-2-carboxamide
4-[1-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
6-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-3-carbonitrile
N-cyclopropyl-3-[5-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
1-(furan-3-ylmethyl)-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1,9-dimethyl-4-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecane
(3S,4S)-1-(5-amino-1H-pyrazole-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-(1-butyl-1H-imidazol-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
3,6,7-trimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
3-(3,5-difluoro-4-methoxyphenyl)-1H-pyrazole
3-(3-methoxyphenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
2-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5-(dimethylamino)-2,3-dihydropyridazin-3-one
3-{[8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyridin-2-amine
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-3-hydroxypyridine-2-carboxamide
2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
[1-({[(2E)-3,7-dimethylocta-2,6-dien-1-yl]amino}methyl)cyclobutyl]methanol
5-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-fluorophenyl)methyl]-N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{[1-(1-butanoylpiperidin-4-yl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridin-2-one
1-[1'-(2H-1,3-benzodioxole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
(1-{[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl]amino}cyclopentyl)methanol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2,2-dimethylpropanoyl)-2,8-diazaspiro[4.5]decan-3-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-sulfonamide
3-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-(4,6-dimethylpyridin-2-yl)-3-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)benzamide
4-methyl-9-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
N-methyl-3-(3-methylphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
2-[(4-chlorophenyl)methyl]-8-methanesulfonyl-2,8-diazaspiro[4.5]decan-3-one
7-hydroxy-6-methoxy-4-(2-methoxypyridin-3-yl)-1,2,3,4-tetrahydroquinolin-2-one
3-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
1-(3,4-dimethylphenyl)-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]({[5-(furan-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})methylamine
3-(4-tert-butylbenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-3-(2-oxopiperidin-1-yl)propanamide
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
N-(2-methylprop-2-en-1-yl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-[4-(hydroxymethyl)phenyl]acetic acid
N-{3-[({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}carbamoyl)methoxy]phenyl}propanamide
2,7,8-trimethyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)quinoline-4-carboxamide
2-(2-methoxyphenyl)-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-4-[2-(furan-2-yl)pyrimidin-5-yl]-7-methyl-5H,7H-thieno[3,4-b]pyridine-3-carbonitrile