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N-(3-chlorophenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
5-methyl-1-(4-methylphenyl)-4-[4-(trifluoromethyl)benzoyl]piperazin-2-one
3-(azepane-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[5-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
[(3R,4R)-1-(6-chloro-2H-chromene-3-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]propan-1-one
N-(2-{[5-chloro-2-(methylamino)phenyl]formamido}ethyl)-2,2,2-trifluoroacetamide
2-[4-(2,3-dihydro-1H-indene-5-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
(2S)-2-amino-3-cyclohexyl-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}propan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl){[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[4-(trifluoromethoxy)phenyl]methyl}acetamide
4-(4-{1-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
4-[2-(1-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]-N,N-dimethylbenzamide
1-(4-methylpiperidin-1-yl)-2-(4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenoxy)ethan-1-one
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[(3,4,5-trimethoxyphenyl)methyl]propanamide
2-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-N,N,4-trimethylpyrimidin-2-amine
3-bromo-5-(pyrrolidine-1-sulfonyl)benzoic acid
2-amino-6-cyclopentyl-5-methyl-4-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}pyridine-3-carbonitrile
1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
3-[2-(dimethylamino)ethyl]-8-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl](isoquinolin-5-ylmethyl)amine
4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2,3,4-tetrahydroquinolin-2-one
N-(1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-chlorobenzamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
2-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propan-1-ol
(3S,4S)-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
(1R,7S)-N-methyl-3-[2-(4-methylphenyl)ethyl]-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1S,5R)-3-(6-chloro-8-methylquinolin-4-yl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N,1-dimethyl-2-oxo-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N3-cycloheptyl-4-oxo-1-(propan-2-yl)-N5-[2-(pyrrolidin-1-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(1,1-dioxo-1λ6-thiolan-3-yl)acetamide
4-{2-[(1-ethyl-3-methylpiperidin-3-yl)formamido]ethyl}benzoic acid
3-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}pyridine
3-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
4-{1-[6-(2-methylpiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
4-(1-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}butan-2-yl)morpholine
2-(1-methyl-1H-pyrazole-5-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-{[(4-methylphenyl)sulfanyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(3-chlorophenyl)-4-(3,5-difluorobenzoyl)-5-methylpiperazin-2-one
(2S,4R)-4-hydroxy-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyrrolidine-2-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(6-methylpyridazin-3-yl)pyrrolidin-3-yl]acetamide
1-(2-methoxyphenyl)-4-{1-[(2-methylphenyl)methyl]piperidin-3-yl}piperazine
N-(2-ethoxyethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-{2-[(dimethyl-1H-1,2,4-triazol-1-yl)methyl]propanoyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-{2-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
2-{1-[(2-ethoxyphenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
4-chloro-N-[(4-hydroxyazepan-4-yl)methyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-(1-butyl-3-methyl-1H-pyrazol-5-yl)-1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]urea