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(3R,9aR)-3-benzyl-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(3R,4S)-1-(furan-2-carbonyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
1-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-3-phenylpropan-1-ol
2-[1-(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
N-benzyl-2-(ethoxymethyl)pyrrolidine-1-sulfonamide
3-(3,4-difluorophenyl)-5-(2-methoxy-3-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
4-(5-methylpyridin-2-yl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-(6-methoxy-3-methyl-1-benzofuran-2-yl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
2-{1-methyl-5-[1-(morpholin-4-yl)cyclohexanecarbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
5-(2-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{2-[(pyridin-3-yl)amino]ethyl}-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
1-{2-[methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})amino]ethyl}cyclopentan-1-ol
4-(2,1,3-benzoxadiazol-5-yl)-1-methyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-methyl-1-(1-{[3-(morpholin-4-ylmethyl)phenyl]methyl}piperidin-4-yl)butan-1-ol
4-[4-(2-methoxyphenyl)benzoyl]-1,2-dimethylpiperazine
N,N,2-trimethyl-7-[1-(4-methylphenyl)cyclopropanecarbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
1-(4-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}phenyl)ethan-1-one
5-(3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-3-yl}phenyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
8-[4-(propan-2-yl)pyrimidin-2-yl]-1-oxa-8-azaspiro[4.5]decan-3-ol
(3R,4R)-4-(hydroxymethyl)-1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]piperidin-3-ol
2-(3-fluorophenyl)-1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidine
N-methyl-4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-2-amine
2-(dimethylamino)-2-(2-methylphenyl)-N-[(2,4,5-trifluorophenyl)methyl]acetamide
2-[(adamantan-1-ylmethyl)({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
N-{[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]methyl}-4-fluorobenzamide
1-[(diethylcarbamoyl)methyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-(1-benzyl-5-{[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]methyl}-1H-1,2,4-triazol-3-yl)acetamide
5-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidin-4-yl}pyridin-2-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(4-methoxyphenyl)methyl](prop-2-yn-1-yl)amine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(oxan-4-yl)azepan-4-amine
N-({3-methyl-7-[2-(naphthalen-2-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(propan-2-yl)acetamide
N-[2-(4-methoxyphenyl)ethyl]-2,5-dimethyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-{3-methyl-2-oxo-2H,3H-imidazo[1,2-a]pyridin-3-yl}acetamide
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
N-[1-(4-methanesulfonylphenyl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(5-ethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-1-(2-chloro-6-fluorobenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
5-[2-(ethylamino)ethyl]-1-(2-phenylpropyl)pyrrolidin-2-one
4-{5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]pyridin-2-yl}thiomorpholine
1,3-dimethyl-2,6-dioxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide