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{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methylphenyl)methyl]amine
2-methoxy-3-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyrazine
1-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}pyrrolidin-2-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-(oxan-2-ylmethyl)acetamide
({3-[(1-cyclohexanecarbonylpiperidin-3-yl)methoxy]phenyl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
3-(2-ethylphenoxy)-1-(3-fluorobenzoyl)azetidine
3-{1-[2-(morpholin-4-yl)butyl]-4-phenyl-1H-imidazol-5-yl}phenol
3-(ethylsulfanyl)-1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]propanamide
(3S,4R)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
7-(2-hydroxyethyl)-2-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(phenylsulfanyl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)spiro[2.2]pentane-1-carboxamide
2-(morpholin-2-yl)-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}ethan-1-one
N-methyl-2-[methyl(phenyl)amino]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
5-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
3-{4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carbonyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
N,2,2-trimethyl-N-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}oxan-4-amine
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
3-methoxy-1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
1-cyclohexyl-N-methyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
1-(cyclohexylmethyl)-6-oxo-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[(propan-2-yl)amino]pyridine-3-carboxamide
1-(azocan-1-yl)-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N,N,4,5-tetramethyl-6-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-2-amine
(1S,5R)-6-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
8-[1-(4-chlorophenyl)cyclobutanecarbonyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
1-cyclohexyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
3-[(4-fluorophenyl)formamido]-N-[3-(propan-2-yloxy)propyl]propanamide
1,3-dimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(5-chloro-2-methylphenyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-(4-chlorophenyl)-2-hydroxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
4-(morpholine-4-carbonyl)-N-[4-(1H-pyrazol-4-yl)phenyl]piperidine-1-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[2-(oxan-4-yl)ethyl]benzamide
3-{5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}-1-methylpyrrolidin-2-one
6-fluoro-2-({[3-(4-methyl-1,3-thiazol-2-yl)propyl]amino}methyl)quinolin-4-ol
7-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
8-(2-propoxyethyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 1-(cyclopropylmethyl)-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-(5-phenoxyfuran-2-carbonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-N,N-dimethylpyrrolidine-2-carboxamide
N-(2-fluorophenyl)-3-{1-[1-(4-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}propanamide
5-(2,3-dihydro-1H-inden-2-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-1-one
N-[(2-fluorophenyl)methyl]-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide