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2-{[1-(1H-indol-1-yl)propan-2-yl]amino}-N-(pyrazin-2-yl)acetamide
N-(1,4-dioxan-2-ylmethyl)-2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methylbenzamide
N-[3-(1H-pyrazol-5-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
7-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
[(3R,4R)-1-[4-(difluoromethoxy)benzoyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(2,3-difluorophenyl)methyl]-5-{2-[(2-phenoxyethyl)amino]ethyl}pyrrolidin-2-one
N-(2-hydroxypropyl)-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
methyl 3-(2-methoxyacetamido)-5-[(oxan-4-yl)amino]-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
6-methyl-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
4-(5-acetylthiophene-3-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-cyclopentyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)oxolane-2-carboxamide
(2S,4S,5R)-2-ethyl-4-[(1-ethylcyclopropyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
N-methyl-3-[(2-methylpyrrolidin-1-yl)sulfonyl]-N-(1,3-thiazol-2-ylmethyl)benzamide
2-(pyridin-4-yl)-N-[3-(pyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide
(2S)-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-3-phenylpropanamide
N-(cyclopropylmethyl)-4-{[(4-methyl-1,3-thiazol-2-yl)methyl]sulfamoyl}benzamide
3-(3,4-dimethoxybenzoyl)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(propan-2-yl)pyrimidine-4-carboxamide
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-3-methylpiperazine
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
6-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
6-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyrazine-2-carboxylic acid
6-[2-(2-ethoxyphenyl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-amino-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(trifluoromethyl)pyrimidine-5-carboxamide
5-(6-hydroxy-1,4-oxazepane-4-carbonyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-{5-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-methoxyphenoxy}-1-(propan-2-yl)piperidine
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
(1S,5R)-6-(morpholine-4-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
6-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
4-chloro-3-[(4,4-difluoropiperidin-1-yl)methyl]-1-methyl-1H-indazole
(3S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-4-yl)methyl]acetamide
1'-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-imidazol-1-yl)butan-1-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(5-ethylfuran-2-yl)methyl]amine
N-cyclobutyl-3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)propanamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylcyclohex-3-ene-1-carboxamide
2-{9-[(4-methylphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
N-[3-(4-{[2-(2-methoxyphenoxy)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methylfuran-3-carboxamide
N-[(5-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
5-acetyl-N-[(1R,2R)-2-(benzyloxy)cyclopentyl]thiophene-3-carboxamide
3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-{[1-(4-oxopentanoyl)piperidin-3-yl]methyl}-4-phenylbenzamide
(2S)-N,N-dimethyl-1-[2-(4-propanamidophenoxy)acetyl]pyrrolidine-2-carboxamide