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1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
4,4,4-trifluoro-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
N-(1-methoxypropan-2-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol
4-(1-butyl-1H-imidazol-2-yl)-1-(4-ethenylbenzoyl)piperidine
(5S)-5-({[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)pyrrolidin-2-one
3-chloro-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-4-fluoro-1-benzothiophene-2-carboxamide
(1S,5R)-6-[2-(1H-imidazol-2-yl)benzoyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-fluorophenyl)-N-({7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-benzoyl-4-[(5-ethylpyridin-2-yl)methyl]piperazine
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-1,3-benzodiazole
(1S,5R)-3-[2-(4,6-dimethyl-1-benzofuran-3-yl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-methyl-1H-pyrazol-5-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-{6-[(2-fluorophenyl)methoxy]-4-[(4-methoxyphenyl)methyl]-3-oxo-1,4-diazepan-1-yl}-2-phenylethane-1,2-dione
(2S)-1-[3-(pyridin-3-yl)propanoyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-(oxan-4-ylmethyl)pyrimidin-2-amine
6-tert-butyl-1-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(4-acetyl-4-phenylpiperidin-1-yl)-1-(morpholin-4-yl)ethan-1-one
2-hydroxy-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-3-(2-methylphenoxy)propanamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
N-[4-(pyrrolidin-1-yl)butyl]imidazo[1,2-a]pyridine-6-carboxamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-methanesulfonylpropan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-methoxypyridin-3-yl)methyl]piperidin-3-ol
1-{4-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]thiophen-2-yl}ethan-1-one
1-[4-(3-{[(adamantan-2-yl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
2-(2-methoxyethyl)-8-[2-(propylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(5-ethylfuran-2-yl)methyl]-4-(2-methoxyethoxy)piperidine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-4-(3-hydroxy-3-methylbutyl)benzamide
1-[5-(cyclopropylmethyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
(1S,6R)-9-{2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(1H-pyrazol-1-yl)butanamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]acetamide
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carboxamide
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-(2-phenylethyl)-1,2,4-oxadiazole
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
methyl 2-{1-[2-(5-fluoro-2-methylphenyl)acetyl]-3-oxopiperazin-2-yl}acetate
N-{1-[(4-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(1H-1,2,3-triazol-1-yl)acetamide
[2-(4-methoxyphenyl)ethyl][(3-methylphenyl)methyl][(1-methylpiperidin-4-yl)methyl]amine
6-ethyl-N4-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-5-methylpyrimidine-2,4-diamine
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,5-dimethylphenyl)urea
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
3-[(1-phenylcyclopentyl)methyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)azetidin-3-ol
(1R,2S)-N1-tert-butyl-N2-[2-(1H-imidazol-4-yl)ethyl]cyclohexane-1,2-dicarboxamide
2-[4-(methylsulfanyl)phenyl]-N-[2-(pyridin-3-yl)ethyl]acetamide
1-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-2-(2-methoxyethyl)piperidine
3-({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)-1λ6-thiolane-1,1-dione