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4-(1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}azetidin-3-yl)pyridine
2-(cyclopropylmethyl)-8-(2,6-dimethylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
6-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(5-fluoro-1H-indol-2-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}propanamide
butyl (1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
4-[(4-fluorophenyl)methyl]-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}propanamide
3-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-(4-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
6-(3,4-difluorophenyl)-2-ethyl-3-methylpyridine
(3R,9aR)-3-benzyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
N-(2-methoxyethyl)-2,5-dimethyl-1-phenyl-N-(pyridin-4-ylmethyl)-1H-pyrrole-3-carboxamide
4-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-oxo-N-phenylbutanamide
6-(oxolan-2-yl)-2-(4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5-propyl-1,3,4-oxadiazole-2-carboxamide
3-(furan-2-yl)-2-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]propan-1-ol
N-[2-(1H-imidazol-1-yl)ethyl]-3-{[(2E)-2-methylbut-2-en-1-yl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
4-{[2-(2-hydroxyethoxy)phenyl]methyl}-5-methyl-1-(4-methylphenyl)piperazin-2-one
7-(3,4-dimethoxyphenyl)-4-[(2-ethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-N,N-dimethylpyridin-2-amine
3-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
(1S,5R)-3-[2-(2-methoxyphenyl)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(cyclopropylmethyl)piperazin-2-yl)ethan-1-ol
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-4-phenylbutane-1,4-dione
2-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
2-[(4-fluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
3-{3-[3-(isoquinolin-1-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-4-carboxamide
1-(oxan-4-yl)-4-[6-(propan-2-yl)pyridin-2-yl]piperazine
N-(1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,3-dimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-(1-cyclopropanecarbonylpiperidin-3-yl)-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclohexyl-3-(cyclopropylmethyl)-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
{3-[(3-methoxyphenyl)methyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl}methanol
N-(3-methylphenyl)-3-{1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}propanamide
3-cyclopropyl-1-phenyl-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
2-{2-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
1-methyl-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
2-benzyl-N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)-1,3-thiazole-4-carboxamide
N,N,7-trimethyl-2-[2-(pyridin-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
1-(4-phenyl-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)ethan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}piperazine
3-chloro-N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
6-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione