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(3R,4R)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-3,4-dimethylpyrrolidin-3-ol
6-(4-methoxy-3-methylphenyl)-9H-purine
2-methyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[(1-ethylcyclopropyl)methyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
3-({[3-(dimethyl-1,2-oxazol-4-yl)propyl]amino}methyl)piperidin-3-ol
ethyl 2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-1,3-oxazole-4-carboxylate
1-[3-(dimethylamino)pyrrolidin-1-yl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)quinoline-2-carboxamide
methyl 5-[2-(6,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazine-1-carboxamide
6-methyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][2-(2,5-dimethylphenoxy)ethyl]methylamine
2-[4-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-2-ol
[4-(2H-1,3-benzodioxole-5-carbonyl)-1,4-oxazepan-6-yl]methanol
6-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyridine-3-carbonitrile
3-cyclopentyl-1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(2E)-3-(furan-2-yl)-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylprop-2-enamide
2-amino-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-4-methyl-1,3-benzothiazole-6-carboxamide
9-(6-aminopyridine-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S,4R)-4-[3-(4-fluorophenyl)benzamido]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidine-2-carboxylate
N-cyclopropyl-3-{[1-(cyclopropylmethyl)piperidin-4-yl]oxy}-4-methoxybenzamide
2-(1-ethyl-1H-pyrazol-4-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]quinoline-4-carboxamide
4-(1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}propanamide
1-(3-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
2-cyclopropyl-4-hydroxy-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}pyrimidine-5-carboxamide
propan-2-yl 8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
2-(1H-indol-3-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[(3R,4R)-3-hydroxy-1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl]pyridine-4-carboxamide
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}but-2-yn-1-one
N-ethyl-5-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
2-(dimethylamino)-N-[(3-hydroxyphenyl)methyl]-N-methyl-2-(2-methylphenyl)acetamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
4-[2-ethyl-7-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholine
1-(3-ethyl-1,2-oxazole-5-carbonyl)-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
1-[(2-fluorophenyl)methyl]-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-one
N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}-2,1,3-benzothiadiazole-4-sulfonamide
1-(cyclohexylmethyl)-6-oxo-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}piperidine-3-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
3-(2-oxoimidazolidin-1-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
1-(cyclopropylmethyl)-3-hydroxy-3-({[(2-hydroxyadamantan-2-yl)methyl]amino}methyl)piperidin-2-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methyl-1H-1,3-benzodiazole-6-carboxamide
2-(dimethylamino)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}acetamide
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}urea
4-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
1-(furan-2-yl)-2-[4-(5-methylpyridin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethane-1,2-dione