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N-[(2-fluorophenyl)methyl]-2-[(furan-3-ylmethyl)amino]acetamide
1-[(2,5-difluorophenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidine-5-carboxylic acid
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-[(2-methylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
6-[2-(4-chlorophenyl)morpholine-4-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-(oxolan-3-ylmethyl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-3-{[4-(1H-imidazol-1-yl)phenyl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-butyl-5-[(4-oxo-3,4-dihydroquinazolin-3-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)-N-propylacetamide
8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]sulfamoyl}-N,N-dimethylbenzamide
(3aS,6aS)-2-(ethanesulfonyl)-5-[(4-methoxy-2-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
4-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-2-fluoro-6-methoxyphenol
(4aR,7aS)-1-(2-methylpropyl)-4-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(2S)-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidine-2-carbonyl]morpholine
4-[(1R)-1-(4-chlorophenyl)ethyl]-3-cyclopropyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(ethylamino)-4-methyl-N-[6-(phenylamino)pyridin-3-yl]-1,3-thiazole-5-carboxamide
3-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[2-(morpholin-4-yl)propyl]-2-phenylpyrimidine-5-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine
4-ethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1,2,3-thiadiazole-5-carboxamide
2-[6-methyl-2-oxo-4-(trifluoromethyl)-1,2-dihydropyridin-1-yl]propanamide
3-(furan-2-ylmethyl)-1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
3-{1-[(4-chlorophenyl)methyl]-1H-pyrazol-5-yl}-1-methyl-1-[2-(oxan-2-yl)ethyl]urea
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(thiophen-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-chloro-2-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenol
N5-[1-(2-chlorophenyl)ethyl]-N6-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[2-(2-amino-9H-purin-6-yl)phenyl]ethan-1-one
4-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-2-methyl-5-propylpyrimidine
2-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
2-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3-methylquinoxaline
8-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(4-acetylphenoxy)-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)ethan-1-one
2-acetyl-8-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
1,7-dimethyl-2-(thiomorpholine-4-carbonyl)-1H-indole
3-fluoro-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzene-1-sulfonamide
1-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(pyridin-2-yl)piperidin-4-ol
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(3-{4-[3-(dimethylamino)propyl]piperazine-1-carbonyl}phenyl)phenol
11-[5-(methoxymethyl)furan-2-carbonyl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}thiomorpholine
3-{4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}propan-1-ol
1-ethyl-N-[(2-methoxyphenyl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-6-(6-aminopyrimidin-4-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one