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2-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
4-cyclopentyl-7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-methyl-6-(1-methylpiperidin-4-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
1-ethyl-6-methyl-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(adamantan-1-yl)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]acetamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
6-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-(4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-2-(methylamino)pyridine-4-carboxamide
2-(furan-2-yl)-5-[5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyrimidine
2-(5-acetylthiophen-3-yl)-1-[4-(benzenesulfonyl)piperazin-1-yl]ethan-1-one
3-[(4-cyclohexylpiperazin-1-yl)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
(2S,4R)-4-amino-N-methyl-1-[4-(thiophen-2-yl)butanoyl]pyrrolidine-2-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
6-methoxy-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(cyclohex-1-en-1-yl)ethyl]benzamide
N,15-dimethyl-9-(5-methylthiophen-2-yl)-N-(1,2-oxazol-3-ylmethyl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)pyridin-2-amine
8-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-6-benzyl-3-(4-fluorobutyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,5R)-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-benzyl-6-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(4-fluorophenyl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
6-methyl-3-[(3-methyl-1H-pyrazol-5-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(4-fluorophenyl)-N-[2-(2-methoxyethoxy)phenyl]piperidine-1-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
N-(3-chloro-4-fluorophenyl)-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propanamide
dimethyl[(5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}furan-2-yl)methyl]amine
1-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,4-diazepane
1-[1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-[2-({[(5-fluoro-1H-indol-2-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-ethyl-2-oxo-1-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[3-(4-methylpiperazin-1-yl)butyl]benzamide
2-cyclopropanecarbonyl-8-(2,6-diaminopyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
1-(azepan-1-yl)-3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propan-1-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
6-{4-[3-(azocan-1-yl)propanoyl]piperazin-1-yl}pyridine-3-carbonitrile
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[4-(1H-pyrazol-1-yl)phenyl]urea
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[3-(morpholin-4-yl)azetidin-1-yl]butan-1-one
(3S,4S)-1-[2-(2-methoxyphenoxy)ethyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-(carbamoylamino)-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
(1R,5R)-6-benzyl-3-(5-methyl-1,3-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[5-({[(4,6-dimethylpyridin-3-yl)methyl]carbamoyl}amino)-2-methoxyphenyl]-2-methoxyacetamide
5-(diethylamino)-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-benzyl-3-(piperidin-4-yl)-1-(quinolin-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N3-(1-benzylpiperidin-4-yl)-N5-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide