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N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-5-fluoro-2-methylbenzene-1-sulfonamide
3-[(4-cyclopentylpyrimidin-2-yl)amino]-N,2-dimethylpropanamide
9-ethyl-1-methyl-4-[(6-methylquinolin-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-[(2-ethylpyrimidin-5-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
1-[(4-chlorophenyl)methyl]-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-3-(1-methyl-1H-indole-6-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-methyl-3-(piperidine-1-carbonyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}-4,5,6,7-tetrahydro-1H-indazole
4-(2-butyl-1H-imidazol-4-yl)-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{2-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
3-[4-(1-cyclohexanecarbonylpyrrolidine-2-carbonyl)piperazin-1-yl]pyrazine-2-carbonitrile
N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
[(3R,4R)-1-(1H-imidazol-2-ylmethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-[2-(benzyloxy)phenyl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
(1S,6R)-3-methyl-4-oxo-N-(4-phenyl-1,2,3-thiadiazol-5-yl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
7-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(propan-2-yl)-2-(4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-chloro-4-fluorobenzoyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-[(3-methoxyphenyl)methyl]-6-oxo-N-propyl-2,7-diazaspiro[4.5]decane-2-carboxamide
3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
N-cyclohexyl-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methylbenzamide
1-{4-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
1-(1,3-benzoxazol-2-ylmethyl)-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
5-methoxy-N-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
1-(2-aminopyrimidin-4-yl)-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-(2-{2-azabicyclo[2.2.1]heptane-2-carbonyl}pyrrolidin-1-yl)-4-methylquinazoline
2-[N-methyl-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanamide
N-ethyl-6-(3-fluorophenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
3-(4-methoxyphenyl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]propan-1-one
1-[1-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)piperidin-3-yl]pyrrolidin-2-one
5-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methoxyphenol
1-(4-methyl-2-{[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]amino}pyrimidin-5-yl)ethan-1-one
4-(3-amino-1H-1,2,4-triazole-5-carbonyl)-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,2,6-trimethyl-N-(propan-2-yl)quinoline-3-carboxamide
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
(4aS,7aR)-1-(3-aminopropanoyl)-4-benzyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
3-(6-methoxypyridin-3-yl)pyridin-2-ol
2-(2-phenylethyl)-8-(9H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-phenyl-1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
6-[(furan-2-ylmethyl)(methyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
7-[2-(pyridin-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-(3-{4-azaspiro[2.5]octan-4-ylmethyl}phenoxy)-3-[cyclohexyl(methyl)amino]propan-2-ol
2-[1-(1-methyl-6-oxopiperidin-3-yl)-4-phenyl-1H-imidazol-5-yl]benzoic acid