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2-(3-chloro-4-fluorophenoxy)-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]ethan-1-one
N-methyl-4-phenoxy-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}butanamide
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
8-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]isoquinoline
N-(4-fluorophenyl)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-amine
4-{3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carbonyl}benzonitrile
3-benzyl-1-(6-methyl-2-propylpyrimidin-4-yl)piperidine-3-carboxylic acid
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
(2R,6R)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
[2-(1H-indazol-3-yl)ethyl](methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-(5-{5-[(methylsulfanyl)methyl]furan-2-yl}-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl)benzoic acid
N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)acetamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(3-methoxypropyl)piperidine
N-(oxolan-3-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-4-(1-methylpiperidin-4-yl)piperidine
1-methyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(5-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
N-methyl-3-(morpholine-4-sulfonyl)-N-(1,3-thiazol-2-ylmethyl)benzamide
2-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,6-dimethylpyrimidin-2-amine
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-3-methoxy-2-methylbenzamide
N-ethyl-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-{[(2-ethoxyethyl)amino]methyl}-6-methylquinolin-4-ol
1-{4-[2-methoxy-4-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(3S)-1-benzylpyrrolidin-3-yl]-6-cyclopropylpyrimidin-4-amine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(3-hydroxypropyl)benzamide
2,5-dioxo-6-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-cycloheptyl-1-(4-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
N-[(3R,4S)-1-(3-methanesulfonamidopropanoyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(1r,4r)-4-{[2-(3-chloro-4-hydroxyphenyl)acetamido]methyl}-N-methylcyclohexane-1-carboxamide
2-methyl-6-(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)pyrimidin-4-ol
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butanamide
5-(2,5-dimethylphenoxymethyl)-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
6-chloro-3-fluoro-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-cyclopropyl-6-[2-(methylsulfanyl)phenyl]pyridazin-3-amine
(2S,4R)-4-amino-N-ethyl-1-{[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}propane-1,3-diol
3-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
1-(2-{[(5-ethyl-1,3,4-oxadiazol-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
3-[1-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]-N-[2-(propan-2-yloxy)phenyl]piperidine-1-carboxamide
(2S,4R)-4-amino-1-[3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-hydroxy-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}acetamide
(3aS,6aS)-2-(cyclopropylmethyl)-5-[3-(1,2-oxazolidin-2-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-8-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
2-{2-[1-(5-propylthiophene-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide