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1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
N-[(3S,4R)-4-(propan-2-yl)-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-yl]methanesulfonamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylpyridin-2-amine
1-(3-chlorophenyl)-5-methyl-4-[3-(pyridin-2-yl)propanoyl]piperazin-2-one
1-[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methoxypyrimidine
1-[2-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)ethyl]pyrrolidin-2-one
N-(2-{6-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}ethyl)acetamide
{7-[4-methyl-6-(methylsulfanyl)quinolin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-[1-(1-tert-butyl-5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]-N-cyclopropylpropanamide
2-(4-methylphenyl)-N-[2-(methylsulfamoyl)ethyl]quinoline-4-carboxamide
4-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)piperidine-4-carbonyl]morpholine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[3-(piperidin-1-yl)propyl]-1,2-oxazole-3-carboxamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N,N-dimethylpyrimidin-4-amine
6-(4-{[4-(pyridin-2-yl)phenyl]methyl}piperazin-1-yl)pyridine-3-carboxamide
methyl 2-{1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-oxopiperazin-2-yl}acetate
5-butyl-1'-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
7-(5-methylthiophen-2-yl)-4-[2-(pyridin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-ethyl-4-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]ethan-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-ethyl-2-methylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl})amine
2-{[2-amino-7-(1-methyl-1H-pyrazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}-N-methylacetamide
methyl 4-oxo-4-[3-(4-phenylbenzoyl)piperidin-1-yl]butanoate
2-hydroxy-4-methyl-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]pentan-1-one
(1S,5R)-3-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4S)-4-cyclopropyl-1-(5-ethyl-2-methylpyrimidin-4-yl)pyrrolidine-3-carboxylic acid
2-[methyl(5-{[3-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}pyrimidin-2-yl)amino]acetic acid
N-(1-propylcyclopropyl)-2-(2,3,4-trifluorophenyl)acetamide
(3R,4R)-1-(5-chloro-3-fluoropyridin-2-yl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
4-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
1-{6-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyridin-2-yl}ethan-1-ol
N-ethyl-5-[(isoquinolin-5-yloxy)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-(propan-2-yl)-1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}benzamide
N-methyl-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}naphthalene-1-carboxamide
2-(3,4-dimethoxyphenyl)-N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
N-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1-(pyrimidin-2-yl)piperidin-3-amine
5-cyano-2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
5-(2,6-dimethoxyphenyl)-N-{[1-(dimethylamino)cyclohexyl]methyl}-1,2,4-triazin-3-amine
1-ethyl-4-({methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1H-pyrrole-2-carbonitrile
(2S,4R)-4-amino-1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-N-methylpyrrolidine-2-carboxamide