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2-(4-{[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenyl)ethan-1-amine
5-methyl-N-[3-(trimethyl-1H-pyrazol-1-yl)propyl]pyrimidin-2-amine
7-[(3,4-dimethoxypyridin-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decane
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[2-({7-acetyl-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]piperidin-2-one
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxan-4-yl)pyridin-2-amine
2-(1-methylpyrrolidin-3-yl)-9-(pyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(morpholin-4-yl)ethyl]acetamide
4-(1H-imidazol-1-yl)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(1-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperidin-2-yl)methanol
6-(2-phenoxyethyl)-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-cyclopropanecarbonyl-7-[(3-ethenylphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-[3-(dimethylamino)pyrazin-2-yl]-3-ethylpiperidine-3-carboxylic acid
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(thiophene-2-sulfonamido)acetamide
3,3-bis(2-methoxyethyl)-1-[4-(1,3-thiazol-4-yl)phenyl]urea
ethyl 1-{1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carbonyl}piperidine-3-carboxylate
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(thiophen-3-ylmethyl)amine
({1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}sulfamoyl)dimethylamine
6-[(5-chloro-2-propoxyphenyl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(4aS,7aR)-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-N-[(2,3-dimethylphenyl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-tert-butyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-oxopyrrolidine-3-carboxamide
N-(3-methyl-1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperidin-4-amine
5-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine
9-ethyl-4-(1H-indazole-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2-methoxyphenyl)-N-[1-({[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
{1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
3-(azepane-1-carbonyl)-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2,6-trimethylpyridine-4-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(3-methoxybenzoyl)piperazine
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
3-{5-[(2-aminopyridin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-{4-[3-(piperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(oxane-4-carbonyl)pyrrolidine-3-carboxylic acid
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-(4-methylpentan-2-yl)piperidin-4-amine
N-(1-methyl-1H-1,2,3-triazol-4-yl)-4-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzamide
1-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazole
2-(2,1,3-benzothiadiazole-4-sulfonyl)-2,8-diazaspiro[4.5]decane
1-(4-ethoxypyrimidin-2-yl)-N,N-diethylpyrrolidin-3-amine
1-cyclobutanecarbonyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(1,1-dioxo-1λ6-thian-4-yl)-3-(4-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
2-{[(3R,4S)-4-cyclopropyl-1-(2-hydroxyacetyl)pyrrolidin-3-yl]amino}pyridine-3-carbonitrile
{2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}urea
4-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}benzoic acid
1-(cyclohexylmethyl)-4-{[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrrolidin-2-one
N-(2-methylpropyl)-4-(methylsulfanyl)-N-(pyridin-2-ylmethyl)benzamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-hydroxy-N-(2-methoxyethyl)-2-methylpyrimidine-5-carboxamide