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4-(1H-pyrazol-3-yl)-1-(1,3-thiazol-2-ylmethyl)piperidine
3-[(3R,4S)-1-(3-chloro-5-fluorobenzoyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
4-{4-[(2E)-2-methylbut-2-en-1-yl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(2-chlorophenoxy)ethyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
3-[({[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}amino)methyl]-1λ6-thiolane-1,1-dione
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
2-[3-(oxolan-3-yl)-5-{pyrazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazol-1-yl]acetic acid
1-(cyclohexylmethyl)-5-[3-(diethylamino)pyrrolidine-1-carbonyl]-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
methyl 6-[(3,5-dimethylphenyl)methyl]-2-(thiomorpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-({[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl](methyl)amino}methyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
(1S,5R)-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-methoxyphenyl)-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
8-(5-ethyl-1,2-oxazole-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-{imidazo[1,2-a]pyrimidine-2-carbonyl}morpholin-3-yl)-N-(pyridin-3-yl)acetamide
3-(4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)pyridine
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-(isoquinolin-5-ylmethyl)-N-methyl-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[3-(thiophen-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
(3S,4S)-4-(naphthalen-2-yl)-1-(1,2-oxazole-3-carbonyl)piperidin-3-ol
(2S,6S)-6-butyl-1-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-(2,6-dimethylpyridine-4-carbonyl)-4-[2-(3-methoxyphenoxy)ethyl]piperazine
1-(1-cycloheptylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
2-ethyl-9-(4-oxo-4-phenylbutyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
3-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
(1S,5R)-3-(5-methyl-1,2-oxazole-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{7-[5-(methoxymethyl)furan-2-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
(1R,9aR)-1-[({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}amino)methyl]-octahydro-1H-quinolizin-1-ol
(3R)-1-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)pyrrolidin-3-ol
2-cyclohexyl-N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]acetamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-(1H-indazol-1-yl)acetamide
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-(3,5-dimethylphenyl)piperazin-2-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(4-ethylphenyl)methyl]piperidin-4-yl}oxy)benzamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-methylpyrimidine-5-carbonyl)piperidin-3-yl]propanoic acid
dimethyl({1-[4-(quinoxalin-2-yl)phenyl]ethyl})amine
2-{1-[(3,4-difluorophenyl)methyl]-4-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
3-({[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
5-hydroxy-N-[(3-methylphenyl)(thiophen-2-yl)methyl]-4-oxo-4H-pyran-2-carboxamide
2-cyclopentyl-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(7-fluoro-4-methylquinolin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
(3R,5R)-N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
3-(3-fluoro-4-methoxyphenyl)-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1H-pyrazole
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylphenyl)methyl]acetamide
2-ethyl-4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]pyridine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide