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N-[2-(4-methoxyphenyl)ethyl]-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-phenoxyethyl)piperidine
6-(1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
9-[(3,4-dichlorophenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
8-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-8-azaspiro[4.5]decane-7,9-dione
N-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(4-fluorophenyl)-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-(4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
[2-(4-aminophenyl)-8-methylquinolin-3-yl]methanol
N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-6-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[6-hydroxy-4-(5-methyl-1,2-oxazole-3-carbonyl)-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
4-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1,2-dihydrophthalazin-1-one
7-(2-propoxybenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({7-chloro-2-[3-(hydroxymethyl)piperidin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)-5-methylthiophene-2-carboxamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
2-[5-(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl]acetamide
(1S,5R)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-({1-methyl-1H-pyrazolo[1,5-a]imidazol-7-yl}formamido)-N-(1,3-thiazol-2-yl)propanamide
6-tert-butyl-2-(2-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-(1-{7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
2-(dimethylamino)-2-(2-methylphenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}[(2-ethylpyrimidin-5-yl)methyl]amine
4-{1-[1-(propan-2-yl)piperidin-4-yl]azetidin-3-yl}pyridine
3-[2-(dimethylamino)ethyl]-8-(pyrazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{4-[3-(piperidin-1-ylmethyl)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
7-(2-methoxyethyl)-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
8-(1-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]propanamide
3-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
4-{3-[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propoxy}benzamide
1-methyl-4-{1H,3H,4H,5H-thiopyrano[4,3-b]indole-8-carbonyl}piperazine-2-carboxylic acid
N-[(3S,4R)-4-propyl-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]methanesulfonamide
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-4-oxo-4H-chromene-2-carboxamide
(1S,5R)-6-[(3,4-difluorophenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(2-fluorophenyl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
(3aS,6aS)-1-methyl-5-{[4-(2-phenylethoxy)phenyl]methyl}-octahydropyrrolo[3,4-b]pyrrole
3-hexyl-8-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(thian-4-yl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine
4-[(5-chlorofuran-2-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
3-(1-butyl-1H-pyrazol-5-yl)-1-[cyclopropyl(4-methylpyridin-2-yl)methyl]urea
2-ethoxy-4-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
2-methoxy-5-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}benzoic acid
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[(5-methylpyrazin-2-yl)methyl]benzamide
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-methyl-4-[3-(2-phenylethyl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]pyridine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide