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3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methyl-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
1-{4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]thiophen-2-yl}ethan-1-one
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-amine
6-methoxy-N-[2-(5-methylfuran-2-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}azepan-3-amine
[(3R,4R)-1-[(3-methyl-1H-indol-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-({5-[(2R)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-propylpiperidine
(2S,4R)-1-[(4-chlorophenyl)methyl]-4-(cyclooctylamino)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
3-(azepane-1-carbonyl)-5-(4-benzylpiperidine-1-carbonyl)-1-(butan-2-yl)-1,4-dihydropyridin-4-one
3-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[(1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
2-(3-hydroxyphenyl)-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]ethan-1-one
(1S,5R)-6-[(3-chloro-4,5-diethoxyphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
4-(hydroxymethyl)-1-[4-(1H-pyrazol-1-yl)benzenesulfonyl]azepan-4-ol
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-4-(1H-1,2,4-triazol-1-yl)butanamide
8-[(3-methylthiophen-2-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-2-(pyridin-4-ylsulfanyl)acetamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}oxane-4-carboxamide
N-[(3-fluorophenyl)methyl]-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-cyclopropanecarbonyl-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methoxy-N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]acetamide
N-methyl-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]furan-2-carboxamide
(1R,5S,6S)-6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-[(prop-2-en-1-yl)amino]benzamide
3,5-difluoro-2-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)pyridine
2-({[(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-[(2-methyl-1,3-oxazol-4-yl)methyl]-8-azabicyclo[3.2.1]octane
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(3-methoxyphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
methyl[2-(oxan-2-yl)ethyl]{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
[(1-cyclopentylpiperidin-4-yl)methyl][(2-fluoro-5-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
2-{[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methoxy}acetamide
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-(3-methoxyphenoxy)ethan-1-one
3-[5-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)imidazo[1,2-a]pyridine-6-carboxamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(1H-pyrazol-1-yl)acetamide
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
1,5-dimethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrrole-2-carboxamide
3-cyclopropyl-N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-[3-(2-methylphenyl)piperidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine
6-(6-methoxypyridin-3-yl)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-methyl-N-(pyridin-3-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-benzyl-3-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
2-{1-[1-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
N-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
N-ethyl-6-oxo-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,6-dihydropyridine-3-carboxamide