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N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-8-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(2,3-dihydro-1H-isoindol-2-yl)-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}acetamide
8-methoxy-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
3-(4-methylphenyl)-1-[7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
2-[(4aR,7aS)-4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
9-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
methyl (1S,3S,3aR,6aS)-3-(2-chloro-3,6-difluorophenyl)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
[(3-chlorophenyl)methyl]({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
(3R,4R)-4-amino-1-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-ol
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
(2S,4S)-4-(4-{[(cyclohexylcarbamoyl)(methyl)amino]methyl}-1H-1,2,3-triazol-1-yl)-N-ethylpyrrolidine-2-carboxamide
3-(3,4-dimethoxybenzoyl)-1-[(2,6-dimethoxyphenyl)methyl]piperidine
(3aS,6aS)-5-[3-(4-fluorophenoxy)propyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzamide
1-[2-(2,2-diphenylethyl)morpholin-4-yl]-2-methylpropan-2-ol
3-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-(2-methylpropyl)-1H-pyrazole
4-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
3-[1-(6-chloro-8-methylquinolin-4-yl)piperidin-3-yl]propanamide
2,3-dimethyl-4-oxo-N-{3-[(propan-2-yl)carbamoyl]phenyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
1-methyl-4-{4-[3-(3-methylphenoxy)azetidine-1-carbonyl]phenyl}piperazine
N-{[(2S,4S)-4-fluoro-1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)pyrrolidin-2-yl]methyl}methanesulfonamide
N-ethyl-2,8-dimethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
3-(azocan-1-yl)-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-(phenoxymethyl)piperidine
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(2-ethylbutyl)piperidine
3-({ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
[(3R,4R)-1-(2-methoxypyridine-3-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-1-(pyridin-3-ylmethyl)piperidin-4-amine
3-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-(2-ethyl-6-methylphenyl)urea
N-[(3-chlorophenyl)methyl]-N-(2-methylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
3-amino-1-[(2-chloro-6-fluorophenyl)methyl]pyrrolidine-3-carboxylic acid
N-hexyl-3-[(3-methoxypyrrolidin-1-yl)sulfonyl]benzamide
N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide
(4aS,7aR)-1-(dimethyl-1,3-oxazole-4-carbonyl)-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}pyridine
{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
(2-{[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](oxolan-2-ylmethyl)amino}ethyl)dimethylamine
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-ethylphenyl)methyl]piperidine
N-cyclopentyl-N'-{3-[(5-methylpyridin-2-yl)amino]propyl}butanediamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
methyl N-[1-({[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}carbamoyl)ethyl]carbamate
(3aR,7aS)-2-[3-(morpholine-4-carbonyl)benzenesulfonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-cyclopropyl-N-(2-hydroxyethyl)-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(2-{1-[2-(benzyloxy)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-(2,3-dihydro-1H-indol-1-yl)-2-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]ethane-1,2-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(3-methoxypropyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
2-methoxy-3-[4-(2-phenoxyethyl)piperazin-1-yl]pyrazine
4-ethyl-1-[(6-methylpyridin-2-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,9aR)-1-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol