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3-fluoro-4-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
(2R,6S)-1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
4-methyl-1-[(4-methylphenyl)methyl]-1,4-diazepan-5-one
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2-phenylethyl)piperidine
1-(cyclohexylmethyl)-6-oxo-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
1-{3-[(4-fluoropiperidin-1-yl)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-(1-methyl-1H-pyrazol-5-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]propanamide
3-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-N-(1,3-thiazol-2-yl)benzamide
ethyl 1-[(7-fluoro-1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-4-carboxylate
1-methoxy-8-[4-(2-methylpropyl)benzoyl]-1,8-diazaspiro[4.5]decan-2-one
(2S,3R)-2-({[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)-3-hydroxybutanamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-oxo-4H-chromene-2-carboxamide
methyl 2-(4-{[4-(3-hydroxyphenyl)piperidine-1-carbonyl]amino}phenoxy)acetate
N-(1,3-dihydroxypropan-2-yl)-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[(1R,3R)-3-aminocyclopentyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
[2-(cyclohex-1-en-1-yl)ethyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-[(3S,4R)-1-benzyl-4-(dimethylamino)piperidin-3-yl]-N-[2-(morpholin-4-yl)ethyl]propanamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2,4-dimethyl-N-(2-methylpropyl)-1,3-thiazole-5-carboxamide
5-fluoro-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(pyrrolidin-1-yl)pyrimidin-2-amine
(3S,4R)-3-benzyl-4-methyl-1-(pyridin-4-ylmethyl)piperidin-4-ol
4-ethyl-1-[1-(2-fluorophenyl)propan-2-yl]-1,4-diazepan-5-one
1-methyl-3-({4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
1-methyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(3-fluorophenyl)methyl]-6-oxo-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
ethyl 4-({[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}amino)piperidine-1-carboxylate
5-(4-benzylpiperidin-1-yl)-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-cycloheptyl-3-{2-[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}urea
methyl 1-[(3S,5S)-1-[(4-chlorophenyl)methyl]-5-(cycloheptylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(1-{2-amino-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-yl)pyrimidin-2-amine
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-(2-phenylethyl)piperidine
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]-4-(trifluoromethyl)pyridine
3-phenyl-1-{1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}propan-1-one
propyl(pyridin-2-ylmethyl)(pyridin-4-ylmethyl)amine
5-cyclopropanecarbonyl-1'-(2,4-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-4-(3,3,3-trifluoropropyl)pyrimidine
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-(4-hydroxyphenyl)ethan-1-one
5-{1-[2-(ethylsulfanyl)ethyl]-4-phenyl-1H-imidazol-5-yl}-2-(2-methoxyethyl)pyrimidine
4-[(2,5-dimethoxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(1S,5R)-3-benzyl-6-(7-methyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-6-ol
1-methyl-2-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
N-ethyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(pyridin-4-ylmethyl)acetamide
6-(pyrrolidin-1-ylmethyl)-4-(1,3-thiazol-2-ylmethyl)-1,4-oxazepan-6-ol
1-[1-(4-benzylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]-2-(phenylsulfanyl)ethan-1-one