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N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpropanamide
6-(4-chlorophenyl)-2-(3-{[(2-hydroxyethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-methyl-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-1-(4-hydroxy-3-methylbenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
6-(2-chlorophenyl)-N-[(3S)-2-oxoazepan-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-(oxolan-3-yl)acetamide
6-(oxolane-2-carbonyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
2-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane
3-(2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-(1H-indol-3-yl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
(benzylsulfamoyl)({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-(1-cycloheptylpiperidin-3-yl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
{5-[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-2-yl}methanol
N-[(1-methylpyrrolidin-3-yl)methyl]-5-phenoxyfuran-2-carboxamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
(2S)-1-{[4-(6-methyl-2-propylpyrimidin-4-yl)phenyl]methyl}pyrrolidine-2-carboxylic acid
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
3-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylpyrimidin-4-amine
8-[(2S)-2-amino-2-cyclopropylacetyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}-1-(pyridin-3-yl)ethan-1-ol
4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-ethyl-1H-pyrazole
3-(4-methoxyphenyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-3-phenylpropanamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}morpholin-2-yl)ethyl]acetamide
2-(azepan-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]acetamide
11-(4-acetylpiperazin-1-yl)-4-[2-(3-chlorophenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-[2-(methylsulfanyl)benzoyl]-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-methyl-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N,1-dimethyl-5-{[2-(4-phenylpiperidin-1-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-ethyl-5-({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-methyl-5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
ethyl 4-({2-[(pyridin-3-yl)amino]ethyl}amino)piperidine-1-carboxylate
6-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indole
(1S,4S)-2-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-2-azabicyclo[2.2.1]heptane
N-[2-(3-methoxyphenyl)-1-{1-[2-(morpholin-4-yl)propanoyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
5-[(4-fluoro-2-methoxyphenyl)methyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-6-(methoxymethyl)pyridine-2-carboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
3-[1-(1-cycloheptylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
(3aR,7aS)-2-{2-[(5-fluoropyrimidin-2-yl)oxy]hex-5-en-1-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-phenylethyl)piperidine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(methylamino)pyridine-3-carboxamide