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7-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}-5-[(3-fluorophenyl)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
ethyl 2-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]amino}acetate
1-(2,3-dihydro-1H-inden-2-yl)-4-(1-methylazepane-2-carbonyl)-1,4-diazepane
2-(5-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(4-methylpentyl)morpholine
6-{2-[(dimethylamino)methyl]phenyl}-N,N-dimethylpyridazin-3-amine
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methoxyethan-1-one
5-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-chloro-2-(1-ethyl-1H-pyrazol-4-yl)-4-(morpholine-4-carbonyl)quinoline
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(6-methylpyridin-2-yl)methyl]benzamide
methyl({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(1H-pyrazol-5-ylmethyl)amine
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(1S,5R)-3-(3-fluoropyridin-2-yl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3,9-diazaspiro[5.6]dodecane
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-4-(1H-pyrazol-4-yl)butanamide
(4aS,8aR)-1-(piperidin-4-ylmethyl)-6-(pyridin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-(propan-2-yl)-1,3-oxazole
methyl 4-[5-methyl-4-(thiomorpholin-4-ylmethyl)-1,3-oxazol-2-yl]benzoate
2-(2-methyl-1,3-thiazol-4-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(1R,2R,6S,7S)-4-(2,6-difluoro-3-methylbenzoyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-2-propoxyacetamide
2-(adamantan-1-yl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]acetamide
7-methoxy-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1H-3-benzazepine
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(ethyl)methylamine
1-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}sulfonyl)azepane
3-{[(3-cyclohexyl-1,2-oxazol-5-yl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
1-[(4-fluorophenyl)methyl]-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-[4-(4-fluorophenyl)butanoyl]-1-(2-methoxyphenyl)piperazin-2-one
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[3-(oxolan-2-yl)propyl]amine
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-chloro-N-{[1-(ethanesulfonyl)piperidin-3-yl]methyl}benzamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
1-(2-{[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}ethyl)piperidin-4-ol
(4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
3-[3-(4-cyclopropanecarbonylphenyl)phenyl]-1H-pyrazole
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-6-methoxyphenol
2-[4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)morpholin-3-yl]acetic acid
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-{[(oxolan-2-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]but-3-en-1-one
1-{3-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxymethyl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
4-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
5-acetyl-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]thiophene-3-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-(1-benzyl-1H-imidazol-2-yl)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidine
4-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)butan-1-ol
3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]propanamide
1-(cyclohexylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(but-2-yn-1-yl)-5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(furan-2-ylmethyl)-1H-pyrazole-3-carboxamide
5-fluoro-1,3-dimethyl-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}-1H-indole-2-carboxamide