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4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]-1-oxaspiro[4.5]decan-2-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-(1H-imidazol-1-ylmethyl)piperidine
3-(2-amino-1,3-thiazol-4-yl)-N-[(2-ethoxypyridin-3-yl)methyl]propanamide
5-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,3-oxazole-4-carboxamide
(2S,4S)-4-amino-1-{2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]acetyl}-N-methylpyrrolidine-2-carboxamide
4-(4-chlorophenyl)-1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]butan-1-one
(3S,4S)-1-{[4-(benzyloxy)-2-methoxyphenyl]methyl}-4-methylpiperidine-3,4-diol
1-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]propyl}-5-methyl-1H-1,2,3,4-tetrazole
(2S,4S)-4-amino-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[3-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetamide
3-(6-methoxypyridin-3-yl)-5-(morpholine-4-sulfonyl)benzoic acid
1-benzyl-5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(2R,4R,6S)-2-phenyl-6-[4-(1H-pyrazol-1-ylmethyl)phenyl]oxan-4-yl]acetamide
N-[(3R,4R)-3-hydroxy-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-4-yl]pyridine-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylcyclohexane-1-carboxamide
2-{2-[(dimethylamino)methyl]-4-(pyridin-3-yl)phenoxy}-N-(2-phenylethyl)acetamide
2-(4-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-(piperidin-1-yl)-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]butan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
4-(2,2-diphenylethyl)-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
(2-methoxyethyl)({2-phenyl-1-[1-(quinoxalin-6-ylmethyl)piperidin-4-yl]ethyl})(pyridin-3-ylmethyl)amine
5-{3-[(2-fluoroethyl)carbamoyl]benzenesulfonamidomethyl}-N-methylfuran-2-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]propanamide
(3aR,5R,6S,7aS)-2-(5-methylthiophene-2-carbonyl)-octahydro-1H-isoindole-5,6-diol
N-ethyl-4-methyl-5-(3-methyl-3-phenylpiperidine-1-carbonyl)-1,3-thiazol-2-amine
4-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
5-{2-[(1-cyclopropylethyl)amino]pyrimidin-4-yl}-2-ethoxybenzoic acid
2-{[1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]oxy}pyrimidine
4-(1,3-benzothiazol-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenol
3-(5-{[(cyclopropylmethyl)sulfanyl]methyl}-3-phenyl-1H-1,2,4-triazol-1-yl)-1λ6-thiolane-1,1-dione
1-(2H-1,3-benzodioxol-5-yl)-2-(4-methanesulfonylphenyl)-1H-imidazole
7-hydroxy-4-[4-(pyridin-2-yl)phenyl]-1,2,3,4-tetrahydroquinolin-2-one
6-methyl-2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}pyridine-3-carboxamide
[3-(2-methoxyethyl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-3-yl]methanol
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-1,3-dimethyl-1H-indole-2-carboxamide
8-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(4-methylphenoxy)-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
N-(cyclohexylmethyl)-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-methyl-6-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]pyridine
N-[(3S,4R)-1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
3-ethyl-4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazin-2-one
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-[3-(1H-pyrazol-1-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
(1S,5R)-3-[3-(4-fluorophenoxy)propyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(azepan-1-yl)ethyl]-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-methoxyphenyl)-4-[2-(2-methoxyphenyl)acetyl]-6-methylpiperazin-2-one
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-{methyl[(4-methylphenyl)methyl]amino}acetamide