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N-cyclopropyl-5-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{[(1S)-1-carbamoyl-3-methylbutyl]amino}-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 3-[6-methyl-5-({[2-(methylsulfanyl)phenyl]formamido}methyl)-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl]benzoate
8-methoxy-N-[2-(1,3-thiazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[2-(3-chlorophenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(3-methoxypropyl)piperidine-3-carboxamide
2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}ethan-1-one
2-(5,6-dimethylpyrimidin-4-yl)-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
1-benzyl-N3-methyl-4-oxo-N5-(prop-2-en-1-yl)-N3-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-(propan-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-(oxane-4-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-1,4-oxazepan-6-ol
3-(4-chloro-2-methylbenzoyl)-1-(2,3,4-trimethoxybenzoyl)piperidine
(2-{2-[2-(4-methoxyphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N,2-dimethyl-N-[3-(1H-pyrazol-1-yl)propyl]-1H-1,3-benzodiazole-4-carboxamide
5-[1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]-N-(pyridin-2-yl)thiophene-2-carboxamide
4-[(1S,2R)-2-[(5-ethylpyrimidin-2-yl)amino]-1-hydroxypropyl]phenol
2-butyl-8-(2-cyclopropylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]acetamide
5,7-dimethoxy-4-[(2E)-pent-2-en-2-yl]-1,2,3,4-tetrahydroquinolin-2-one
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-(3-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
1-cyclopentyl-5-oxo-N-[2-(pyridin-4-yl)ethyl]pyrrolidine-3-carboxamide
2-[3-(4-fluorophenyl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-cyclohexyl-N-[(3,4-dimethoxyphenyl)methyl]oxolane-3-carboxamide
(2R,4R)-4-hydroxy-N-{2-[3-(trifluoromethyl)phenyl]ethyl}pyrrolidine-2-carboxamide
ethyl 2-{2-[(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazol-4-yl)formamido]ethyl}-1,3-thiazole-4-carboxylate
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(quinolin-4-ylmethyl)amine
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]benzamide
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
1-[4-(3-chloropyridin-2-yl)piperazin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-2-(pyrrolidin-1-yl)acetic acid
(1R,5S,6R)-3-{[2-(difluoromethoxy)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
6-[(3,5-dimethoxyphenyl)methoxy]-4-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1-(propan-2-yl)-1,4-diazepan-2-one
2-(3-phenylpropyl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]morpholine
1-[3-(4-fluorophenyl)phenyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
1-[(8-methoxy-2H-chromen-3-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
3-(morpholine-4-sulfonyl)-5-(thiophen-3-yl)benzoic acid
4-chloro-3-[3-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1H-pyrazol-5-amine
(1S,5R)-3-(4-methylpyrimidine-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(2-oxoimidazolidin-1-yl)benzamide
2-[3-(2,4-dimethoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
[(4-fluoro-3-methoxyphenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
3-hydroxy-3-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)methyl]-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-methoxy-5-{1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
2-(morpholin-3-yl)-N-{3-[(trifluoromethyl)sulfanyl]phenyl}acetamide
N-[3-(furan-2-yl)-3-phenylpropyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
5-ethyl-3-{[2-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
2-(cyclohex-1-en-1-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one