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3-(3-methylbutyl)-8-(1-propanoylpyrrolidine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-2-ethyl-N-(furan-2-ylmethyl)butanamide
3-butyl-1-methyl-4-(3-phenoxypropanoyl)piperazin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-{1-[(1-{spiro[2.4]heptane-1-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}pyridine
dimethyl({[4-methyl-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
2-(azocan-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
3-({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)sulfamoyl)-N-(oxolan-3-ylmethyl)benzamide
3-[(cyclohexylamino)methyl]-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
N5-cyclopentyl-N6-[2-(pyridin-3-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
N-cyclopentyl-3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
(2S,4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-N-ethyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
2-butyl-4-methyl-3-oxo-N-(2-phenylethyl)piperazine-1-carboxamide
1-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[(dimethylamino)methyl]azepan-4-ol
4-methyl-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrimidin-2-amine
1-(furan-2-carbonyl)-4-(piperidine-1-sulfonyl)-1,4-diazepane
4-{3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(2-methylpropyl)piperidin-4-amine
4-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
6-methoxy-3-{[methyl(2-methylpropyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(2-oxopyrrolidin-1-yl)propanamide
1-[2-methoxy-4-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
(4aR,8aR)-2-methanesulfonyl-7-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-decahydro-2,7-naphthyridin-4a-ol
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-ethyl-N-methyl-5-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-yl}-2-phenylethan-1-one
3-phenyl-1-(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-1-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
5-fluoro-2-[1-(4-methyl-1H-imidazole-5-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]benzamide
2-[benzyl({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amino]ethan-1-ol
(3S,4R)-4-(2-methoxyphenyl)-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidine-3-carboxylic acid
2-(morpholin-4-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-cyclopropyl-N-[2-(morpholin-4-yl)butyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-methylpyridine-3-carboxamide
(3R,9R)-11-(2,3-difluorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
(3S,5S)-1-(2-methylpropyl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-1,2-dihydroquinolin-2-one
4-benzyl-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[6-(dimethylamino)pyridine-3-carbonyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{4-[(3-methoxyphenyl)methyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl}methanol
1-[(2-fluorophenyl)methyl]-4-[2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-[(3R,4S)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]oxane-4-carboxamide