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2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2-methoxyphenoxy)-1-(morpholin-4-yl)ethan-1-one
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-N-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-methyl-5-oxo-1-(pyridin-3-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxamide
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
4-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]-2-methylphenol
5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine-2,4-diol
6-ethyl-N-{[1-(3-methylphenyl)pyrrolidin-3-yl]methyl}pyrimidin-4-amine
1-methyl-2-oxo-8-(quinoline-6-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(2S,4S)-4-acetamido-N-ethyl-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidine-2-carboxamide
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(cyclobutylmethyl)(oxolan-2-ylmethyl)amine
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
1-methyl-5-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-oxazepane
1-[4-(piperazine-1-sulfonyl)benzoyl]piperidin-3-ol
2-{5-[3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,4-diazepan-5-one
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperazine
4-(piperidin-1-yl)-6-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidine
ethyl 4-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
6-{[(1-ethylpyrrolidin-2-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
9-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
[(2S,6S)-4-[4-(propan-2-yl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N4-{1-oxaspiro[4.4]nonan-3-yl}-6-(propan-2-yl)pyrimidine-2,4-diamine
1-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}acetamide
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
7-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-({3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}methyl)propanamide
N-[4-(2-methoxy-2-phenylacetamido)phenyl]-5-methylfuran-2-carboxamide
N-(2-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}ethyl)acetamide
N-cyclopentyl-3-[5-(pyridine-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
{5-[4-(ethylamino)pyrimidin-2-yl]-2-fluorophenyl}methanol
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-4-(cyclopropylmethyl)piperazine
1-methyl-5-(2-methylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-2-[4-(1-methyl-1H-imidazol-2-yl)-1H-pyrazol-1-yl]acetamide
3-phenyl-1-(5-phenyl-1,2-oxazole-4-carbonyl)piperazine
N-benzyl({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}amino)sulfonamide
2-methoxy-3-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
1-(1H-indazol-7-yl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]propan-1-one
{1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol
2-(1-methyl-4-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-2-yl)ethan-1-ol
8-(6-aminopyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
8-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-8-azaspiro[4.5]decane-7,9-dione
3-(4-methyl-1H-pyrazol-5-yl)-1-[2-(trifluoromethyl)benzenesulfonyl]piperidine
ethyl 2-{4-[3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanoyl]morpholin-3-yl}acetate
3-(1H-pyrazol-1-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide