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(2H-1,3-benzodioxol-5-ylmethyl)({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})methylamine
N-[3-(dimethylamino)propyl]-N-methyl-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-amine
1-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}ethan-1-one
1-(4-methylpiperazin-1-yl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-[2-(3-methoxyphenyl)ethyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
N-[1-(4-ethyl-3,3-dimethylpiperazin-1-yl)-1-oxopropan-2-yl]methanesulfonamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[4-(isoquinolin-5-yl)-1H-pyrazol-1-yl]-N-methylacetamide
2-methyl-N-[2-(pyridine-2-sulfonyl)ethyl]thieno[2,3-d]pyrimidin-4-amine
5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole
2-methyl-6-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
[(3R,4R)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-chloro-5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}azepane
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
2-methyl-3-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}quinoxaline
N-({7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)ethane-1-sulfonamide
4-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
2-(pyridin-2-ylmethyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
[(2S,6S)-4-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[(3-methyl-1H-indol-2-yl)methyl]amine
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(3,4-difluorophenyl)propanamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}cyclopropanesulfonamide
4-[(2S)-1-(7-methyl-1-benzofuran-2-carbonyl)pyrrolidine-2-carbonyl]morpholine
4-(4-phenoxybutyl)-1,2-dihydropyridin-2-one
4-[(4-methylphenyl)sulfanyl]-1-(pyrrolidin-3-ylmethyl)piperidine
[1-(3-chlorobenzoyl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl]acetamide
N-({1-[(4-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-amino-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-6-(2,4-dimethoxybenzoyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2,3-dihydro-1H-isoindole
2-(dimethylamino)-N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-2-(4-methylphenyl)acetamide
2-methyl-N-(1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{[3-(1H-pyrazol-5-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
N-[(2,6-difluoro-3-methylphenyl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
3-(5-methyl-2,1,3-benzothiadiazol-4-yl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
(1S,5R)-3-(2-ethylpyrimidine-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-imidazol-1-yl)propan-1-one
N-({3-[3-(hydroxymethyl)phenyl]phenyl}methyl)acetamide
9-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(2-methoxyethyl)(methyl)amino]-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[3-(furan-2-yl)phenyl]-N-[4-(methylamino)butyl]piperidin-4-amine
4-({5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)oxane-4-carbonitrile
N-{3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]propyl}pyridin-3-amine
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[2-(1H-pyrazol-1-yl)phenyl]methyl}amine
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(quinolin-4-yl)pyrrolidin-3-amine
2-(dimethylamino)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,4-dimethylpyrimidine-5-carboxamide