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9-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidin-4-amine
1-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(propan-2-yl)urea
(1S,5R)-6-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
4-benzyl-2-{2-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-{[3-(cyclopentyloxy)phenyl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
9-[(2,5-dimethylphenyl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-benzyl-5-[5-(thiophen-2-yl)-1H-pyrazol-4-yl]-1H-1,2,4-triazole
(4aS,8aR)-6-(4-methylpyrimidine-5-carbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-(3-{[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
4-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
1-ethyl-3-methyl-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-2-[(4-chlorophenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(azocan-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-chloro-N-(1,4-dioxan-2-ylmethyl)-4-fluoro-1-benzothiophene-2-carboxamide
4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-7-fluoro-2-methylquinoline
1-ethyl-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
3-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2,2-dimethylpropan-1-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(1,3-dihydroxypropan-2-yl)piperidine-3-carboxamide
3-[5-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
2-{4-[4-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-6-methylpyrimidin-2-yl}phenol
3-(4-fluorophenoxymethyl)-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
1-(furan-2-ylmethyl)-N-[1-(2-phenylethyl)piperidin-3-yl]piperidine-4-carboxamide
7-[2-(methylamino)pyrimidine-5-carbonyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
5-[1-(2-methoxyacetyl)pyrrolidin-2-yl]-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]thiophene-2-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]pyrrolidin-3-yl]methanol
4-(1H-1,3-benzodiazol-1-yl)-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine-4-carboxylic acid
1-{4-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
1-{4-[3-cyclopropyl-5-(pyridin-2-yl)-1H-1,2,4-triazol-1-yl]phenyl}-N-methylmethanesulfonamide
(1S,4S)-2-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
N,6,6-trimethyl-5-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}thiomorpholine-3-carboxamide
methyl (2S,4R)-4-(4-fluorobenzamido)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxylate
5-methyl-N4-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrimidine-2,4-diamine
N2-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-(pyridin-3-yl)pyrazine-2,3-diamine
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-butylpyridine-2-carboxamide
8-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(4-tert-butylphenoxymethyl)-5-(morpholin-2-ylmethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-(3-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
1-methyl-3-(2-methylpropyl)-N-{[1-(pyridin-2-yl)piperidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
7-(3-chlorophenyl)-4-(pyrimidin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{3-[ethyl(methyl)amino]propyl}-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-ethyl-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
2-(dimethylamino)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-({5-[(5-fluoro-2-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-(4-acetylphenoxy)-1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}ethan-1-one
8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine